STRATEGY FOR SELECTIVE REDUCTIVE ADDITION
D. Chusov, Russian Academy of Sciences, Moscow, Russia
DIVERGENT SYNTHESIS OF NATURAL SESQUITERPENE LACTONES: ONE PLAN, MANY PITFALLS TO AVOID
A. Zografos, Aristotle University of Thessaloniki, Thessaloniki, Greece
TOTAL SNTHESIS OF POLYCYCLIC NATURAL PRODUCTS
Th. Magauer, University of Innsbruck, Innsbruck, Austria
RECENT DEVELOPMENTS IN LOW PRESSURE CARBONYLATIONS
T. Skrydstrup, Aarhus University, Aarhus, Denmark
TRANSFER OF REACTIVE GASES FROM ONE MOLECULE TO ANOTHER
M. Oestreich, Technische Universität Berlin, Berlin, Germany
DONOR–ACCEPTOR OLIGOPYRROLES
M. Stępień, University of Wrocław, Wrozław, Poland
THE FINE BALANCE BETWEEN STABILITY AND ENZYMATIC DEGRADABILITY OF POLYMERIC CARRIERS - THE IMPORTANCE OF MOLECULAR PRECISION
R. Amir, Tel-Aviv University, Tel-Aviv, Israel
TRAPPING OF REACTIVE INTERMEDIATES
J. Roithova, Radboud University, Nijmegen, The Netherlands
DISCOVERY OF THE FIRST ANTIBACTERIAL AGENT INHIBITING THE ENERGY-COUPLING FACTOR (ECF) TRANSPORTERS BY STRUCTURE-BASED VIRTUAL SCREENING
A.K.H. Hirsch, Saarland University, Saarbrücken, Germany
COUNTER-ION MEDIATED APPROACHES TO CONTROLLING AXIAL CHIRALITY
M.D. Smith, University of Oxford, Oxford, UK
INTERACTION VS. FRUSTRATION IN BIMETALLIC COOPERATIVE SYSTEMS
J. Campos, Universidad de Sevilla, Sevilla, Spain
TARGETING BACTERIAL PERSISTERS IN THE POST-ANTIBIOTIC ERA
S. Sattin, Università degli Studi di Milano, Milan, Italy
NECESSITY IS THE MOTHER OF INVENTION: NATURAL PRODUCTS AND THE CHEMISTRY THEY INSPIRE
S.E. Reisman, California Institute of Technology, Pasadena, USA
RECENT ADVANCES TO ACCESS FLUORINATED SCAFFOLDS
T. Besset, Normandie Université, Rouen, France
HYBRID DISCOVERY WORKFLOW FOR ORGANIC MATERIALS AND SUPRAMOLECULAR SELF-ASSEMBLIES
R. Greenaway, University of Liverpool, Liverpool, United Kingdom
EXPANDING THE BILE ACID CHEMICAL SPACE: SYNTHETIC STRATEGIES FOR LEAD DISCOVERY AND DEVELOPMENT
A. Gioiello, Universita di Perugia, Perugia, Italy
TOTAL SYNTHESIS OF AVENAOL VIA ASYMMTRIC O-ALKYLATION USING CHIRAL AMMONIUM SALT
Y. Takemoto, Kyoto University, Kyoto, Japan
LOW-VALENT Bi(I)⇄Bi(III) REDOX CATALYSIS
J. Cornella, Max-Planck-Institut für Kohleforschung, Mülheim/Ruhr, Germany
NOVEL REACTIONS VIA ELECTROPHILIC ENOLONIUM SPECIES
A. Szpilman, Ariel University, Ariel, Israel
REACTION PROGRESS KINETIC ANALYSIS BY DIRECT ANALYSIS OF CONCENTRATION-TIME PROFILES
R. Pollice, ETH Zürich, Zürich, Switzerland
A TOP-DOWN APPROACH TO DIVERSE LEAD-LIKE SCAFFOLDS
C. Townley, University of Leeds, Leeds, United Kingdom
DEVELOPMENT AND SCALE-UP OF CONTINUOUS FLOW PROCESSES FOR THE MANUFACTURE OF ACTIVE PHARMACEUTICAL INGREDIENTS
P. Poechlauer, Thermo Fisher Scientific, Linz, Austria
DESIGNING NEW SYNTHETIC CONCEPTS FOR IMPARTING MOLECULAR COMPLEXITY WITH C-1 SOURCES
V. Pace, University of Vienna, Vienna, Austria
THE SYNTHESIS AND OPTIMISATION OF NEW ANTIBIOTICS
A. Abell, University of Adelaide, Adelaide, Australia
RATIONAL DESIGN OF NEW, MORE POTENT ACRIDINIUM VISIBLE LIGHT ORGANO-PHOTOCATALYSTS BY C-H FUNCTIONALIZATION
O. García Mancheño, University of Münster, Münster, Germany
ORGANO- AND BIOCATALYSIS FOR LIGNAN NATURAL PRODUCT SYNTHESIS
M. Lazzarotto, University of Graz, Graz, Austria
CHEMO-DIVERGENT NICKEL(0)-CATALYZED ARENE C-F ACTIVATION WITH ALKYNES: UNPRECEDENTED DOUBLE-INSERTION
L. Capdevila, Universitat de Girona, Girona, Spain
SYNERGISTIC CATALYSIS IN DONOR-ACCEPTOR CYCLOPROPANE CHEMISTRY
D.B. Werz, TU Braunschweig, Braunschweig, Germany
GOLD-CATALYZED CROSS-COUPLING-TYPE REACTION OF BROMOALKYNES WITH ALLYLSILANES THROUGH A CONCEALED REARRANGEMENT
M. Zanini, Institute of Chemical Research of Catalonia (ICIQ), Tarragona, Spain
SEQUENTIAL MULTI-BOND FORMING REACTIONS APPLIED TO THE SYNTHESIS OF CONFORMATIONALLY RESTRICTED MDM2-p53 INHIBITORS SUITABLE FOR INTERMITTENT DOSING
A. Gollner, Boehringer Ingelheim RCV GmbH and Co KG, Vienna, Austria
ENANTIOSELECTIVE FRIEDEL-CRAFTS ALKYLATION RECTION OF TRIFLUOROMETHYLATED N-H KETIMINE WITH HETEROARENES BY MEANS OF CHIRAL PHOSPHORIC ACID
T. Akiyama, Gakushuin University, Tokyo, Japan
DYNAMIC CARBON ISOTOPE EXCHANGE OF PHARMACEUTICALS WITH LABELED CO2
D. Audisio, Université Paris-Saclay, Gif-sur-Yvette, France
ACCESS TO UNUSUAL HETEROCYCLIC COMPOUNDS UTILIZING A KEY COBALT-CATALYZED C-H FUNCTIONALIZATION APPROACH
Ch.J. Whiteoak, Sheffield Hallam University, Sheffield, UK
4-π-PHOTOCYCLISATION OF DIHYDROPYRIDAZINES: ACCESS TO VERSATILE BICYCLIC DIAZETIDINES
S. Coote, Lancaster University, Bailrigg, UK
MACROCYCLIC ANION CARRIERS
H. Valkenier, Université libre de Bruxelles, Bruxelles, Belgium
CONTROLLING THE CIRCADIAN CLOCK WITH HIGH TEMPORAL RESOLUTION THROUGH PHOTODOSIMETRY
D. Kolarski, University of Groningen, Groningen, The Netherlands
1,2-DIOXANES AS POTENTIAL ANTI-LEISHMANIAL DRUGS
A. Quintavalla, University of Bologna, Bologna, Italy
THE HUNT FOR ARTIFICIAL REACTIVITIES IN BIOCATALYSIS: FUNGAL COPPER-DEPENDENT METALLOPROTEINS AS MEDIATORS FOR PERICYCLIC REACTIONS
J. Deska, Aalto University, Espoo, Finland
N-NITROHETEROCYCLES: EASILY ACCESSIBLE, BENCH-STABLE AND BROADLY APPLICABLE NITRATING REAGENTS
D. Katayev, Swiss Federal Institute of Technology, Zürich, Switzerland
STORAGE OF INFORMATION USING SMALL ORGANIC MOLECULES
M.J. Fink, Harvard University, Cambridge, USA
QUEST FOR ASYMMETRIC KULINKOVICH REACTION: FROM MECHANISM TOWARDS ENHANCED ENANTIOSELECTIVITY
D. Kananovich, Tallinn University of Technology, Tallinn, Estonia
CONCISE TOTAL SYNTHESES OF (–)-JORUNNAMYCIN A AND (–)-JORUMYCIN ENABLED BY ASYMMETRIC CATALYSIS
E. Welin, California Institute of Technology, Pasadena, USA
SURPRISES WITH ALKYNES: A NEW REACTIVITY PARADIGM AND ITS APPLICATIONS
A. Fürstner, Max-Planck-Institut für Kohleforschung, Mülheim/Ruhr, Germany
MAKING NEW FORMS OF NANOCARBONS
K. Itami, Nagoya University, Nagoya, Japan
TRANSLATIONAL CHEMISTRY
Ph.S. Baran, Scripps Research, La Jolla, USA
ORIGINS OF LIFE SYSTEMS CHEMISTRY
J.D. Sutherland, MRC Laboratory of Molecular Biology, Cambridge, UK
ENANTIOSELECTIVE CATALYSIS OF PHOTOCHEMICAL REACTIONS
Th. Bach, Technical University Munich, Garching, Germany
PEPTIDE DRUGS FROM NATURE – STRUCTURAL AND (BIO)SYNTHETIC ASPECTS OF NEW ANTIBIOTICS
R.D. Süssmuth, Technical University of Berlin, Berlin, Germany
LEWIS ACID ENABLED NOVEL REACTIVITIES IN ASYMMETRIC COPPER CATALYSIS
S.R. Harutyunyan, University of Groningen, Groningen, The Netherlands
ORGANIC SYNTHESIS IN THE EXCITED STATE
P. Melchiorre, Institut Català d’Investigació Química (ICIQ), Tarragona, Spain
FLUORINE CHEMISTRY FOR APPLICATIONS IN MEDICINE
V. Gouverneur, University of Oxford, Oxford, UK
RADICAL CHEMISTRY IN THE DESIGN AND SYNTHESIS OF ARTIFICIAL MOLECULAR MACHINES
J.F. Stoddart, Northwestern University, Illinois, United States
CARBOXYLATES AS DIRECTING AND LEAVING GROUPS IN CATALYTIC BOND FORMATION
L.J. Gooßen, Ruhr-Universität Bochum, Bochum, Germany
INHIBITION STUDIES ON A PANEL OF HUMAN CARBONIC ANHYDRASES WITH N1-SUBSTITUTED SECONDARY SULFONAMIDES INCORPORATING THIAZOLINONE OR IMIDAZOLONE-INDOLE TAILS
F.M. Awadellah, Cairo University, Cairo, Egypt
SYNTHESIS, ANTI-PROLIFERATIVE ACTIVITY AND 2D-QSAR STUDY OF SOME 8-ALKYL-2,4-BISBENZYLIDENE-3-NORTROPINONES
R. George, Cairo University, Cairo, Egypt
SYNTHETIC STUDIES OF NOVEL SPIRO PYRAZOL-3-ONES CONTAINING QUINAZOLINE AND/OR OXIRANE MOIETY
H. Nagabuchi, Fukuoka University, Fukuoka, Japan
REGIOSELECTIVE C-H ARYLATION OF NITRO HETEROCYCLES AND FURTHER TRANSFORMATION OF MANIPULABLE NITRO GROUP
V. Iaroshenko, Polish Academy of Sciences, Łodź, Poland
PREPARATION OF VINYL BORONIC ESTERS VIA A HOMOLOGATION REACTION: BIDIRECTIONAL SYNTHESIS OF MACHILLENE
J. Fordham, University of Bristol, Bristol, UK
TAMING AMBIDENT TRIAZOLE NUCLEOPHILES: REGIOSELECTIVE ION-PAIRING AND PHASE-TRANSFER ORGANOCATALYSIS
H. Dale, The University of Edinburgh, Edinburgh, UK
TOTAL SYNTHESIS OF α-TOCOPHEROL THROUGH ENANTIOSELECTIVE IRIDIUM-CATALYZED FRAGMENTATION OF A SPIRO-CYCLOBUTANOL INTERMEDIATE
F. Ratsch, University of Cologne, Cologne, Germany
UNUSUAL SECONDARY KINETIC ISOTOPE EFFECTS IN REACTION OF TERTIARY PHOSPHINES WITH ELECTRON-DEFICIENT ALKENES
A. Salin, Kazan Federal University, Kazan, Russia
DEVELOPMENT OF ORGANIC POLYMER DONOR FOR EFFICIENT TERNARY ORGANIC SOLAR CELLS
I.H. Jung, Kookmin University, Seoul, Republic of Korea
SYNTHESIS OF AXIALLY CHIRAL BIS(BIBENZYLS) DERIVED FROM PERROTTETIN E VIA C-H ACTIVATED HECK TYPE CYCLIZATION
L. Marx, Saarland University, Saarbrücken, Germany
SULFOXIDE CONTROLLED SUZUKI C-C COUPLING FOR THE SYNTHESIS OF CYCLOPHANE TYPE AXIALLY CHIRAL BIARYLS
S. Bauspieß, Saarland University, Saarbrücken, Germany
PALLADIUM-CATALYZED SEQUENTIAL ARYLATION OF CYCLIC VINYLOGOUS ESTERS
Y.-C. Yang, National Chiao Tung University, Hsinchu, Taiwan
LIGNIN VALORIZATION BY COBALT-CATALYZED FRACTIONATION OF LIGNOCELLULOSE TO YIELD MONOPHENOLIC COMPOUNDS
D. Di Francesco, Stockholm University, Stockholm, Sweden
INTRAMOLECULAR INTERACTIONS IN [2.2]PARACYCLOPHANES
L.M. Birsa, Alexandru Ioan Cuza University of Iasi, Iasi, Romania
TRICYCLIC FLAVONOIDS WITH 1,3-DITHIOLIUM SUBSTRUCTURE: SYNTHESIS AND ANTIBACTERIAL ACTIVITY
L.G. Sarbu, Alexandru Ioan Cuza University of Iasi, Iasi, Romania
DEVELOPING A 'REVERSE-BIOMIMETIC' SYNTHESIS OF AROGENATE AND ITS ANALOGUES
L. Eagling, University of Bristol, Bristol, UK
ASYMMETRIC ORGANOCATALYSIS - SYNTHESIS OF CYCLOHEPTA[B]INDOLES BY (4+3) CYCLOADDITION
G. Levitre, Université Paris-Saclay, Gif-sur-Yvette, France
TRANSFER HYDROCYANATION OF α- AND α,β-SUBSTITUTED STYRENES CATALYZED BY BORON LEWIS ACIDS
P. Orecchia, Technische Universität Berlin, Berlin, Germany
ENANTIOSELECTIVE SYNTHESIS OF HYPERFORIN
S. Frey, Saarland University, Saarbrücken, Germany
STEREOSELECTIVE SYNTHESIS OF NATURAL MYRTUCOMMULONES
T. Jung, Saarland University, Saarbrücken, Germany
ENANTIOSELECTIVE SYNTHESIS OF PROPARGYL ALCOHOLS WITH DIYNES UNDER CARREIRA CONDITIONS
D. Trenz, Saarland University, Saarbrücken, Germany
CONCISE SYNTHESIS OF ALL-CIS-3,4,5-SUBSTITUTED PIPERIDINES THROUGH CASCADE RADICAL CYCLISATION INITIATED BY VISIBLE LIGHT-PROMOTED HYDROSILYLATION OF ALKENES
Z.-J. Yao, Nanjing University, Jiangsu, China
CHEMOSELECTIVITY IN PERHYDROLYSIS OF KETONES, KETALS, AND EPOXIDES
Y. Wu, Chinese Academy of Sciences, Shanghai, China
BASE-CATALYZED STEREOSPECFIC ISOMERIZATION OF ALLYLIC HALIDES
V. García-Vázquez, Stockholm University, Stockholm, Sweden
PHOTOREDUCIBLE Au(III) COMPLEXES FOR CATALYSIS
B. Bibal, Université de Bordeaux, Talence cedex, France
REARRANGEMENT OF 1,2,3-BENZOTHIADIAZINES
I. Gyűjtő, Budapest University of Technology and Economics, Budapest, Hungary
SUPRAMOLECULAR SELF-ASSEMBLY OF HALOGEN-BOND-FORMING QUINOLINE DERIVATIVES
J. Alfuth, Gdansk University of Technology, Gdansk, Poland
NEW POTENT STEROID SULFATASE (STS) INHIBITORS BASED ON FLUORINATED 4-(1-PHENYL-1H-[1,2,3]TRIAZOL-4-YL)-PHENYL SULFAMATES. SYNTHESIS AND BIOLOGICAL EVALUATION
K. Biernacki, Gdansk University of Technology, Gdansk, Poland
SYNTHESIS AND ANTIFUNGAL ACTIVITY STUDY OF TRIMETHYL LOCK-MODIFIED GLUCOSAMINE-6-PHOSPHATE SYNTHASE INHIBITOR
M. Nowak, Gdansk University of Technology, Gdansk, Poland
SYNTHESIS OF 2,4-DIAMINOPYRIMIDINES AS POTENTIAL ANTIFOLATES
A.L. Rousseau, University of the Witwatersrand, Johannesburg, South Africa
DEVELOPMENT OF AMPHIPATHIC CELL-PENETRATING FOLDAMERS FOR DELIVERY OF BIOMACROMOLECULES
T. Misawa, National Institute of Health Sciences, Kanagawa, Japan
PALLADIUM CATALYZED N-ARYLATION OF 1H-TETRAZOLE-5-AMINES
A. Nikolic, University of Belgrade, Belgrade, Serbia
RHODIUM-CATALYSED (3+1+2) CYCLOADDITIONS OF ELECTRON-POOR CYCLOPROPANES
A. Dalling, University of Bristol, Bristol, UK
BIFUNCTIONAL AMINO-REAGENTS FOR C-N BOND FORMATION
J. Farndon, University of Bristol, Bristol, UK
N-HETEROCYCLIC CARBENE-CATALYZED CONCERTED NUCLEOPHILIC AROMATIC SUBSTITUTION OF ARYL FLUORIDES BEARING α,β-UNSATURATED CARBONYL MOIETY
K. Yasui, Osaka University, Osaka, Japan
SYNTHESIS OF A CHONDROITIN SULFATE PROBE AND ITS APPLICATION IN PROSTATE CANCER CELLS
M. Viera, National University of Singapore, Singapore, SIngapore
BIOMIMETIC HALOGENATIONS AT UNACTIVATED C-H BONDS
T. Ambrosio, GSK Carbon Neutral Laboratories for Sustainable Chemistry, Nottingham, UK
C6’-SULFATED CHONDROITIN SULFATE (CS-C) DISACCHARIDE AND TETRASACCHARIDE THROUGH A SHORT SYNTHESIS ROUTE
Y.S. Chng, National University of Singapore, Singapore, SIngapore
CHIRAL AND NON CHIRAL N-BOC PROTECTED 7-AZAINDOLINES IN BATCH AND FLOW
A. Porzelle, Apollo Scientific Ltd., Cheshire, UK
AMIDO-GROUPS AS REMOVABLE DIRECTING GROUPS IN PALLADIUM CATALYZED CARBON-HYDROGEN BOND FUNCTIONALIZATION OF BENZOQUINONE DERIVATIVES
F.-E. Hong, National Chung Hsing University, Taichung, Taiwan
MULTI-CATALYTIC ENANTIOSELECTIVE METHODOLOGY AS ENTRY TO NEW SUPRAMOLECULAR TOOLS
A. Quintard, Aix-Marseille Université, Marseille, France
ASYMMETRIC BIOCATALYTIC PICTET-SPENGLER REACTION TO SHORTCUT ORGANIC SYNTHESIS
W. Kroutil, University of Graz, Graz, Austria
VISIBLE-LIGHT ENABLED LATE-STAGE AMINOCARBONYLATION OF ALKYL IODIDES WITH CARBON MONOXIDE
M. Sardana, AstraZeneca, Gothenburg, Sweden
CONSTRUCTION OF HETEROGENEOUS CATALYSTS AND DYNAMIC INTERFACES ON A POLYDOPAMINE PLATFORM
A. Kunfi, Hungarian Academy of Sciences, Budapest, Hungary
NITRENE-BASED N-N BOND FORMATION: AN EFFICIENT METHOD TOWARDS NITROGEN-RICH TRICYCLIC TRIAZAPENTALENES
E. Pasquinet, CEA, Monts, France
CONTROLLED REDUCTION OF CARBOXAMIDES TO ALDEHYDES, ALCOHOLS OR AMINES
D.Y. Ong , Nanyang Technological University, Singapore, Singapore
DEMYSTIFYING THE SOAI REACTION
S. Athavale, University of Illinois, Urbana, United States
STUDIES TOWARDS THE TOTAL SYNTHESIS OF ASADANIN
J. Ongouta, Symrise AG, Holzminden, Germany
100 G TO 1 KG - THE FORGOTTEN SCALE?
A. Porzelle, Apollo Scientific Ltd., Cheshire, UK
TOWARDS THE TOTAL SYNTHESIS OF CRENARCHAEOL
M. Holzheimer, Rijksuniversiteit Groningen, Groningen, The Netherlands
HIGHLY ENANTIOSELECTIVE DEAROMATIZATION OF PYRYLIUM DERIVATIVES WITH A HELICAL MULTIDENTATE ANION-BINDING CATALYST
M. Gómez-Martínez, University of Münster, Münster, Germany
SELECTIVE FUNCTIONALIZATION OF CYCLIC IMIDES AND AMIDES WITH RUTHENIUM CATALYSTS
Y.-C. Yuan, Université de Rennes 1, Rennes, France
STABLE AND REUSABLE Pd-BNPs CATALYSED STEREOSELECTIVE SYNTHESIS OF (E)-3-ALKYLIDENE OXINDOLES
N. Parveen, Indian Institute of Technology Madras, Chennai, India
1,2-ZWITTERIONIC Ga COMPLEXES OF METHYLIDENEMALONATES AND THEIR REACTIONS WITH ACETYLENES
D. Borisov, Russian Academy of Sciences, Moscow, Russia
ENABLING FRAGMENT GROWTH WITH PHOTOREDOX CATALYSIS THROUGH HIGH-THROUGHPUT EXPERIMENTATION
B. Cons, Astex Pharmaceuticals, Cambridge, UK
CASCADE RADICAL CYCLISATION ON ALKYNYL VINYLOGOUS CARBONATES FOR THE DIVERGENT SYNTHESIS OF TETRASUBSTITUTED FURANS AND DIHYDROFURANS
. Padmaja, Indian Institute of Technology Bombay, Mumbai, India
ONE-POT ALKENE HYDROBORATION/MIGRATORY SUZUKI-MIYAURA CROSS-COUPLING
Y. Baumgartner, University of Basel, Basel, Switzerland
AN ANION-DIRECTED APPROACH TO ENANTIOENRICHED α-TRIARYL AMINES
M. Gredicak, Rudjer Boskovic Insitute, Zagreb, Croatia
UNLOCKING NATURES CHEMICAL TREASURE TROVE - NOVEL NATURAL PRODUCTS FROM MICROBIAL SYMBIONTS
Ch. Beemelmanns, Hans-Knöll Institute (HKI), Jena, Germany
C-C CROSS COUPLING OF TRITYL RADICALS: REACTIVITY AND SPIN DENSITY DELOCALIZATION
N. Fleck, Universität Bonn, Bonn, Germany
MULTICOMPONENT ORGANOCATALYTIC SYNTHESIS OF ISOXAZOLIDIN-5-ONES
J. Annibaletto, Normandie Université, Rouen, France
DFT STUDY OF THE REACTIVITY OF TRANSIENTLY GENERATED CYCLIC DIENOLATES VERSUS THE ACYCLIC COUNTERPARTS IN ADDITION REACTIONS
G. Zanella, Universidad del País Vasco, San Sebastián, Spain
CONTROLLED RELEASE OF MICELLE PAYLOAD VIA SEQUENTIAL ENZYMATIC AND BIOORTHOGONAL REACTIONS IN LIVING SYSTEMS
K. Porte, Université Paris-Saclay, Gif-sur-Yvette, France
RECENT ADVANCES IN "ONLY" GOLD-CATALYZED PHOTOCHEMISTRY
S. Witzel, Heidelberg University, Heidelberg, Germany
ISOTHIOUREA-CATALYSED REGIOSELECTIVE ACYLATIVE KINETIC RESOLUTION OF AXIALLY CHIRAL BIARYL DIOLS
S. Qu, University of St. Andrews, St. Andrews, Scotland
DIVERGENT COBALT-MEDIATED FORMAL (2+2+3)-CYCLOADDITION OF ENEDIYNES: EXPERIMENTAL AND THEORETICAL INSIGHTS
L. Commeiras, Aix-Marseille Université, Marseille, France
STEREOSPECIFIC α-SIALYLATION BY SITE-SELECTIVE FLUORINATION
T. Hayashi, Westfälische Wilhelms-Universität Münster, Münster, Germany
TETHER-DIRECTED REGIOSELECTIVE SYNTHESIS OF AN EQUATORIALFACE BISADDUCT OF AZAFULLERENE USING CYCLO-[2]-OCTYLMALONATE
N. Chronakis, University of Cyprus, Nicosia, Cyprus
SYNTHESIS OF PYRRAZOLE AND PYRIMIDINE STRUCTURE
L. Hammal, University of Science and Technology Houari Boumediene (USTHB), Algiers, Algeria
A BIO-INSPIRED POLYCYCLIZATION OF DIEN-N-YNES DRIVEN BY VISIBLE LIGHT
G. Maestri, Università di Parma, Parma, Italy
SYNTHESIS OF 2,4-DISUBSTITUTED 9,9’-SPIROBIFLUORENES AND FLUORO DISPIROINDENO[2,1-C]FLUORENES THROUGH CATALYTIC [2+2+2] CYCLOTRIMERIZATION
I. Caivano, Charles University of Prague, Prague, Czech Republic
PHOTOREDOX / NICKEL-CATALYZED CARBAMOYLATION OF (HETERO)ARYL BROMIDES
N. Alandini, Institut Català d’Investigació Química (ICIQ), Tarragona, Spain
INTERMOLECULAR CATALYST TURNOVER IN ENANTIOSELECTIVE AMMONIUM ENOLATE CATALYSIS: A SYNTHETIC AND MECHANISTIC STUDY
C. McLaughlin, University of St. Andrews, St. Andrews, Scotland
HIGHLY EFFICIENT SYNTHESIS OF TRISUBSTITUTED PYRAZOLES AND DISUBSTITUTED ISOXAZOLES VIA INTRAMOLECULAR WITTIG REACTIONS: A DIVERSITY-ORIENTED SYNTHESIS OF HETEROARENE SCAFFOLDS
P. Khairnar, National Taiwan Normal University, Taipei, Taiwan
DIVERGENT TOTAL SYNTHESIS OF (+)-EPICOCCIN G AND (-)-ROSTRATIN A ENABLED BY DOUBLE C(sp3)-H ACTIVATION
P. Thesmar, University of Basel, Basel, Switzerland
MECHANISTIC INVESTIGATION OF AN OXIME ETHER ELECTROCYCLIZATION
L. Sotorrios, University of the Basque Country, Donostia/San Sebastian, Spain
AN INTRAMOLECULAR CYCLOADDITION APPROACH TO THE KAURANOID FAMILY OF DITERPENE METABOLITES
B. Callebaut, Ghent University, Ghent, Belgium
AQUA REGIA IN GOLD(III) CHEMISTRY
V. Levchenko, University of Oslo, Oslo, Norway
PARADIGMS OF COOPERATIVE VS. NON-COOPERATIVE LIGANDS IN METAL PINCER COMPLEXES IN (DE)HYDROGENATION REACTIONS
M.H.G. Prechtl, Roskilde Universitet, Roskilde, Denmark
SYDNONE-BASED APPROACH TO HETEROHELICENES THROUGH 1,3-DIPOLAR-CYCLOADDITIONS
E. Yen-Pon, Université Paris-Saclay, Gif-sur-Yvette, France
THE REVISED MECHANISM OF COPPER-FREE SONOGASHIRA CROSS-COUPLING REACTION
M. Gazvoda, University of Ljubljana, Ljubljana, Slovenia
GENERATING AND EXPLOITING SULFINYL NITRENES
Th. Davies, University of Oxford, Oxford, UK
INTRA- AND INTERMOLECULAR STEREOSELECTIVE [2+2] CYCLOADDITION REACTIONS OF ETHENETRICARBOXYLATES AND STYRENES
S. Yamazaki, Nara University of Education, Nara, Japan
NEW DIRECTIONS IN THE HETARENE N-OXIDES CHEMISTRY
L. Fershtat, N.D. Zelinsky Institute of Organic Chemistry, Moscow, Russia
BIOMIMETIC SITE- AND ENANTIOSELECTIVE C–H OXYGENATION OF QUINOLONE ANALOGUES MEDIATED BY HYDROGEN BONDING
F. Burg, Technical University Munich, Garching, Germany
BICYCLIC β-LACTAM INTERMEDIATES FOR THE DIVERGENT SYNTHESIS OF MARINE POLYCYCLIC GUANIDINIUM ALKALOIDS
A. Ribaucourt, NC State University, Raleigh, USA
OXIDANT-FREE Au(I)/Au(III) C-HETEROATOM CROSS-COUPLING CATALYSIS
X. Ribas, Universitat Autònoma de Barcelona, Bellaterra, Spain
SYNTHESIS AND BIOCHEMICAL EVALUATION OF AN ARTIFICIAL, FLUORESCENT GLUCOSINOLATE (GSL)
P. Klahn, Technical University of Braunschweig, Braunschweig, Germany
GOLD-TRIGGERED DEAROMATIZATION CASCADES
E. Van der Eycken, Katholieke Universitei Leuven, Leuven, Belgium
SYNTHESIS OF MULTI RING-FUSED PEPTIDOMIMETICS INTERACTING WITH α-SYNUCLEIN FIBRILS
D. Adolfsson, Umeå University, Umeå, Sweden
ZIRCONIUM IN THE CROWN. ENANTIOSELECTIVE ALKENYLATION OF ALDEHYDES WITH PROTECTED PROPARGYLIC ALCOHOLS IN THE PRESENCE OF CROWN ETHER: A NOVEL APPROACH TO THE INHIBITION OF ACHIRAL BACKGROUND REACTIONS
T. Bauer, University of Warsaw, Warsaw, Poland
DESIGN, SYNTHESIS AND EVALUATION OF NOVEL ∆2-THIAZOLINO 2-PYRIDONE DERIVATIVES AS MYCOBACTERIUM TUBERCULOSIS TOLERANCE INHIBITORS
S. Sarkar, Umeå University, Umeå, Sweden
SINGLE C–F BOND CLEAVAGE OF TRIFLUOROMETHYLARENES WITH A LATENTLY TRANSFORMABLE ORTHO-SILYL GROUP
S. Yoshida, Tokyo Medical and Dental University (TMDU), Tokyo, Japan
BORYL RADICAL MEDIATED LIGNIN DEGRADATION: DEPOLYMERIZATION AND RECONECTION
L. Hong, Justus Liebig University Giessen, Giessen, Germany
CATALYTIC C—C/C—H ACTIVATION RELAY: SYNTHESIS OF NAPHTHOQUINOLIZINIUM SALTS FROM 1-AZABIPHENYLENE
M. Kotora, Charles University of Prague, Prague, Czech Republic
SIMPLIFYING THE SYNTHESIS OF VIRGINIAMYCIN MII ANALOGUES FOR CRYO-EM GUIDED DRUG DEVELOPMENT
L. Scott, Monash University, Melbourne, Australia
STEREOSELECTIVE AND MODULAR ASSEMBLY METHOD FOR DAUCANE, CYATHANE AND TIGLIANE TERPENOID SCAFFOLDS
M. Christiaens, Ghent University, Ghent, Belgium
RADICAL CHEMISTRY OF POLYMER-SUPPORTED DIAZIDOIODATE(I)
T. Kösel, Leibniz University Hannover, Hannover, Germany
DEVELOPMENT OF A TOTAL SYNTHESIS OF CEBULACTAMS A1 AND A2
H. Berneaud-Kötz, Leibniz University Hannover, Hannover, Germany
IMPROVED SYNTHESIS OF CYSTOBACTAMID 861-2 AND ANALOGS
M. Moeller, Leibniz University Hannover, Hannover, Germany
REGIOSELECTIVE CHLORINATION OF IMINOSYDNONE FOR ULTRAFAST CLICK AND RELEASE
M. Feng, Université Paris-Saclay, Gif-sur-Yvette, France
SYNTHESIS OF BODIPY HETERODIMER FORMED BY HYDROGEN BONDING FOR ELECTRONIC TRANSFER INVESTIGATIONS
M. Cordaro, Università di Messina, Messina, Italy
RADIOISOTOPE-ENABLED TRACKING OF SUBSTRATES IN SUZUKI CROSS-COUPLING REACTION
L. Rejc, University of Ljubljana, Ljubljana, Slovenia
1H–15N HMBC NMR AS A TOOL FOR RAPID IDENTIFICATION OF AZAINDOLE CANNABINOID DRUGS
B.A. Martek, University of Ljubljana, Ljubljana, Slovenia
CATALYTIC FORMATION OF C-S BONDS
I. Fleischer, University of Tübingen, Tübingen, Germany
DUAL-CATALYTIC TRANSITION METAL SYSTEMS FOR FUNCTIONALIZATION OF UNREACTIVE SITES OF MOLECULES
D. Lichosyt, University of Strasbourg, Strasbourg, France
ISOMERIZATION IN METATHESIS REACTIONS: UNDESIRED SIDE PROCESS OR USEFUL TRANSFORMATION
A. Kajetanowicz, University of Warsaw, Warsaw, Poland
THE SYNTHESIS OF β,β-DISUBSTITUTED ALLYL ALCOHOLS AND THEIR TRANSFORMATION INTO UNNATURAL AMINO ACIDS
A. Narczyk, Polish Academy of Science, Warsaw, Poland
STUDIES TOWARDS THE TOTAL SYNTHESIS OF HETEROCLITIN F AND TAIWANSCHIRIN A, B, C AND D
M. Haughey, University of Oxford, Oxford, UK
NICKEL CATALYZED REDUCTIVE DEAMINATIVE ARYLATION AT sp3 CARBON CENTERS
R. Martin-Montero, Institute of Chemical Research of Catalonia (ICIQ), Tarragona, Spain
C-C BOND ACTIVATION INITIATED CASCADE PROCESSES
O. Sokolova, University of Bristol, Bristol, UK
DINICKEL OXIDATIVE ADDITION COMPLEXES IN C-O CLEAVAGE: RELEVANCE IN CATALYTIC C–Si BOND-FORMATION
R.J. Somerville, Institute of Chemical Research of Catalonia (ICIQ), Tarragona, Spain
LEWIS BASE-CATALYZED REARRANGEMENTS OF ELECTRON-POOR CYCLOPROPANES
S. Xu, Xi’an Jiaotong University, Xi’an, China
PHOSPHINE-CATALYZED ACTIVATION OF ALKYLIDENECYCLOPROPANES: REARRANGEMENT TO FORM POLYSUBSTITUTED FURANS AND DIENONES
X. He, Xi’an Jiaotong University, Xi’an, China
REGIOSPECIFIC N-ARYLATION OF ALIPHATIC AMINES UNDER MILD AND METAL-FREE REACTION CONDITIONS
G. Kervefors, Stockholm University, Stockholm, Sweden
COMPUTATIONAL INVESTIGATIONS INTO ENANTIOSELECTIVE SAMARIUM DIIODIDE-MEDIATED RADICAL CYCLISATION REACTIONS
N. Beattie, University of Manchester, Manchester, United Kingdom
TRANSCRIPTION OF SELF-ASSEMBLED GEL NETWORKS EMBEDDED WITH REACTIVE VINYL GROUPS TO NANOSTRUCTURED POLYMERS
L. Frkanec, Ruđer Bošković Institute, Zagreb, Croatia
NEW BENCH-STABLE ALLYLATION REAGENTS - HOW TUNING THE REACTIVITY ENABLES HIGHLY ENANTIOSELECTIVE ACCESS TO ALL STEREOISOMERS OF TERTIARY HOMOALLYLIC ALCOHOLS
M. Mantel, Heinrich-Heine-University Düsseldorf, Jülich, Germany
COMPUTATIONAL "DIVE" INTO A NICKEL(0)-CATALYZED ARENE C-F ACTIVATION WITH ALKYNES
S. Roldan-Gomez, Universitat de Girona, Girona, Spain
SITE-SELECTIVE CARBONYLATIVE ROUTES TO FUSED POLYHETEROCYCLIC STRUCTURES
N. Della Ca', Università di Parma, Parma, Italy
A GENERAL HYDROCYANATION OF ACTIVATED TERMINAL ALKYNES
D. Tejedor, Instituto de Productos Naturales y Agrobiología, Tenerife, Spain
STRAIGHTFORWARD SYNTHESIS OF α-AMINO NITRILES THROUGH Mo(CO)6 -CATALYZED REDUCTIVE FUNCTIONALIZATION OF CARBOXAMIDES
P. Trillo, Umeå University, Umeå, Sweden
METAL-FREE REGIOSELECTIVE C-H ARYL-ARYL CROSS-COUPLING - ARYLATION OF 2-NAPHTHOLS WITH DIARYLIODONIUM SALTS
M. Ghosh, University of Warsaw, Warsaw, Poland
REGIOSELECTIVE DISILYLATION OF ALLENES BY DIHYDROSILANE CATALYZED BY GOLD NANOPARTICLES
M. Kydonakis, University of Crete, Heraklion, Greece
SYNTHESIS OF NOVEL LIPID I AND LIPID II ANALOGS
L.M. Wingen, University of Bonn, Bonn, Germany
STUDIES TOWARDS THE TOTAL SYNTHESIS OF TUSCORON C
S. Spindler, University of Bonn, Bonn, Germany
ANOMERIC CONTROL FOR TREHALOSE TRANSFERASE
L. Mestrom, Delft University of Technology, Delft, The Netherlands
A VERSATILE KETONE FORMATION VIA HIGHLY ACTIVE PRECATALYST "POXAP": APPLICATION TO THE SYNTHESIS OF ISOPREKINAMYCIN
F. Bihel, Université de Strasbourg, Illkirch, France
CYSTEINE–SPECIFIC DUAL LABELLING OF PROTEINS USING STRAINED [2.2.1]AZABICYCLIC VINYL SULFONES
A.J. Moreno-Vargas, Universidad de Sevilla, Sevilla, Spain
EVIDENCE FOR TRIPLET SENSITIZATION IN THE VISIBLE-LIGHT-INDUCED [2+2]-PHOTOCYCLOADDITION OF ENIMINIUM IONS
F.M. Hörmann, Technical University Munich, Garching, Germany
IODONIUM SALTS AS GROUP TRASFER REAGENTS - N-HETEROCYCLIC CARBENE-CATALYZED SYNTHESIS OF VINYL AND PROPARGYL KETONES
A. Rajkiewicz, University of Warsaw, Warsaw, Poland
ARYLAZO SULFONES: PHOTOACTIVATABLE SUBSTRATES FOR METAL-FREE ARYLATIONS
S. Protti, University of Pavia, Pavia, Italy
MECHANISTIC STUDIES ON OXIDATIVE DEAROMATIZATION OF PHENOLS PROMOTED BY HYPERVALENT IODINE SPECIES
K. Kraszewski, University of Warsaw, Warsaw, Poland
SEMISYNTHESIS OF NOVEL MACROLIDE-BASED ANTIBIOTICS
S. Heinrich, Ruhr-Universität Bochum, Bochum, Germany
CATALYTIC CLEAVAGE OF C(sp2)-C(sp2) BONDS WITH METAL-CARBYNOIDS
L. Jiang, Institute of Chemical Research of Catalonia (ICIQ), Tarragona, Spain
STEREOSELECTIVE ADDITIONS TO ALKYNES BY IRON AND COBALT CATALYSTS
A. Jacobi von Wangelin, University of Hamburg, Hamburg, Germany
SYNTHESIS AND APPLICATIONS OF VINYL TRIAZENES
A. Suleymanov, Ecole Polytechnique Federale de Lausanne (EPFL), Lausanne, Switzerland
GOLD-PROMOTED ANTI-MARKOVNIKOV HYDROTHIOLATION OF OLEFINS USING EX SITU GENERATED METHANETHIOL
S.K. Kristensen, Aarhus University, Aarhus, Denmark
NEW ACCESS TO PLANAR BLATTER RADICALS: π EXTENDED HETEROCYCLES WITH HIGH SPIN DELOCALIZATION
P. Bartos, University of Lodz, Lodz, Poland
SYNTHESIS AND INVESTIGATION OF Ag-NHC COMPLEXES WITH CYTOTOXIC PROPERTIES TOWARDS CELL LINES MODELLING ACUTE MYELOID LEUKEMIA
F. Lundevall, University of Bergen, Bergen, Norway
TOTAL SYNTHESIS AND BIOLOGICAL EVALUATION OF PELOFEN, A NEW MICROTUBULE-STABILIZING AGENT
J. Van der Eycken, Ghent University, Ghent, Belgium
PALLADIUM-CATALYZED TANDEM ISOMERIZATION/HYDROTHIOLATION OF ALLYL ARENES
P.M. Kathe, University of Tübingen, Tübingen, Germany
VINYLOGY CONCEPT IN THE SYNTHESIS OF SELECTED CARBO- AND HETEROCYCLES
Ł. Albrecht, Lodz University of Technology, Lodz, Poland
RATIONAL DESIGN OF COOPERATIVITY IN A SYNTHETIC RECEPTOR
M. Rondelli, Instituto de Productos Naturales y Agrobiología, San Cristóbal de La Laguna, Spain
REUSABLE POLYSTYRENE-SUPPORTED ORGANOCATALYSTS
I. García-Monzón, Instituto de Productos Naturales y Agrobiología, San Cristóbal de La Laguna, Spain
SYNTHESIS OF NEW PHARMACOLOGICALLY ORIENTED NO-DONOR FUROXAN-BASED HETEROCYCLIC ENSEMBLES
N. Makhova, Russian Academy of Sciences, Moscow, Russia
INTEGRATIVE PERICYCLIC CASCADE: AN ATOM ECONOMIC, MULTI C-C BOND-FORMING STRATEGY FOR THE CONSTRUCTION OF MOLECULAR COMPLEXITY
S. Delgado-Hernandez, Instituto de Productos Naturales y Agrobiología, Tenerife, Spain
C5-DISUBSTITUTED MELDRUM’S ACID DERIVATIVES AS PLATFORM FOR THE ORGANOCATALYTIC SYNTHESIS OF C3-ALKYLATED DIHYDROCOUMARINS
J.-F. Brière, Normandie Université, Rouen, France
CYCLOTRIMERIZATION OF NUCLEOBASE-LINKED NITRILES FOR THE PRODUCTION OF NOVEL S-TRIAZINES
J. Elaridi, Lebanese American University, Beirut, Lebanon
TOTAL SYNTHESIS OF INDOLE ALKALOIDS
T. Szabó, Egis Pharmaceuticals PLC, Budapest, Hungary
SYNTHESIS OF DOUBLE NO-DONORS INCORPORATING FUROXAN AND AZASYDNONE RINGS
E. Zhilin, N.D. Zelinsky Institute of Organic Chemistry, Moscow, Russia
SYNTHESIS OF FUNCTIONALIZED BENZOFURANS FROM PARA-QUINONE METHIDES VIA PHOSPHA-1,6-ADDITION/O-ACYLATION/WITTIG REACTION
Y.-C. Liou, National Taiwan Normal University, Taipei, Taiwan
DOUBLE VINYLOGOUS REACTIVITY OF THE γ AND γ' POSITIONS OF CYCLIC 2-ENONES: ORGANOCATALYSED ASYMMETRIC SYNTHESIS OF FUSED CARBOCYCLES
G. Vassilikogiannakis, University of Crete, Heraklion, Greece
BASE-CATALYZED ISOMERIZATION OF DIENYL ALKYL ETHERS AND DIENOLS: DFT STUDIES
A. Carretero-Cerdán, Stockholm University, Stockholm, Sweden
ORGANOCATALYTIC [3+2]-ANNULATIONS OF β,γ-UNSATURATED-γ-LACTAMS WITH α,β-UNSATURATED ALDEHYDES
M. Sofiadis, University of Crete, Heraklion, Greece
NEW METHODS OF DIRECT CATALYTIC ALKELENATION OF HETEROCYCLES
M. Hachem, Normandie Université, Rouen, France
2-SUBSTITUTED dATP DERIVATIVES AS BUILDING BLOCKS FOR ENZYMATIC SYNTHESIS OF DNA MODIFIED IN THE MINOR GROOVE
J. Matyašovský, Academy of Science of the Czech Republic, Prague, Czech Republic
SYNTHESIS OF NOVEL HETERO-FUSED 7-DEAZAPURINE RIBONUCLEOSIDES
L. Veselovska, Academy of Science of the Czech Republic, Prague, Czech Republic
DEAROMATIZATION OF ELECTRON POOR ARENES BY (4+2) CYCLOADDITION REACTION
B. Rkein, Normandie Université, Rouen, France
NEW METHOD FOR THE SYNTHESIS OF (N-FUROXANYL)HYDRAZONES
D. Bystrov, Russian Academy of Sciences, Moscow, Russia
Ru(II) COMPLEXES CONTAINING EXTENDED π-CONJUGATION BIPYRIDYL ANCILLARY LIGAND: SYNTHESIS AND APPLICATION FOR DSSCs
M. Jeong, Kwangwoon University, Seoul, Korea
DEALING WITH CYCLIZATION IN THE SYNTHESIS OF SPIROINDOL(EN)INES AND TETRAZOLE-ISOQUINOLONES/PYRIDONES HYBRID
G.M. Ojeda, University of Leuven, Leuven, Belgium
INTRAMOLECULAR (4+3) CYCLOADDITIONS OF THIOPHENES
Y. Zheng, The University of Hong Kong, Hong Kong, P.R. China
MORPHOLOGICAL CHANGES OF ORGANIC PHOTOVOLTAICS: MOLECULAR DYNAMICS SIMULATION STUDIES
J. Na, Kwangwoon University, Seoul, Korea
RADICAL MIGRATION FOR SYNTHESIS OF MEDIUM-SIZED RINGS
Z.-L. Li, Southern University of Science and Technology, Shenzhen, China
ORGANOCATALYTIC ASYMMETRIC SYNTHESIS OF ATROPISMERIC BIARYLS
S. Xiang, Southern University of Science and Technology, Shenzhen, China
C-H BOND-INVOLVED INTRAMOLECULAR ASYMMETRIC RADICAL CYCLIZATION
L. Ye, Southern University of Science and Technology, Shenzhen, China
SYNTHESIS AND REACTIVITY OF ALKYNYL VYNIL HYDRAZINES
R. Diana, Instituto de Productos Naturales y Agrobiología, Tenerife, Spain
MECHANISTIC INSIGHTS INTO THE SILYL-PRINS REACTION
L. Evans, University of Greenwich, Chatham Maritime, U.K.
HIGHLY REACTIVE DIENOPHILES FOR BIOORTHOGONAL TETRAZINE LIGATIONS
M. Wilkovitsch, TU Wien, Vienna, Austria
RECENT ADVANCES IN HETEROCYCLIC SYNTHESIS IN AstraZeneca ONCOLOGY
S. Pearson, AstraZeneca, Macclesfield, United Kingdom
TOTAL SYNTHESIS OF CALLYSPONGIOLIDE
B. Wölfl, Max-Planck-Institut für Kohleforschung, Mülheim/Ruhr, Germany
HYDRODIFLUOROMETHYLATION OF ALKENES WITH DIFLUOROACETIC ACID
C.F. Meyer, University of Oxford, Oxford, UK
ENANTIOSELECTIVE SYNTHESIS OF CHIRAL SULFONES BY BASE METAL-CATALYZED ASYMMETRIC CROSS-COUPLING REACTION
D. Qian, Ecole Polytechnique Federale de Lausanne (EPFL), Lausanne, Switzerland
THE ACID-CATALYSED SYNTHESIS OF 7-AZAINDOLES FROM 3-ALKYNYL-2-AMINOPYRIDINES AND THEIR ANTIMICROBIAL ACTIVITY
T. Leboho, University of the Witwatersrand, Johannesburg, South Africa
STEREOSELECTIVE TOTAL SYNTHESIS OF ASPERGILLIDE A
J.B. Mateus-Ruiz, Universidad Nacional Autónoma de México, Ciudad de México, México
CHEMICAL REGENERATION OF AMINE SOLVENTS USING CALCIUM HYDROXIDE FOR CO2 CAPTURE PROCESS
S.K. Jeong, Korea Institute of Energy Research, Daejeon, Korea
PHOTOELECTROCATALYTIC ARENE C-H AMINATION
L. Zhang, Ecole Polytechnique Federale de Lausanne (EPFL), Lausanne, Switzerland
REGIOSELECTIVITY IN BIOCATALYTIC O-METHYLATION OF CATECHOLS
S. Pompei, University of Graz, Graz, Austria
PHOTOCATALYTIC SYNTHESIS OF γ-LACTONES FROM ALKENES: HIGH RESOLUTION MASS SPECTROMETRY AS A TOOL TO STUDY PROTOREDOX REACTIONS
I. Triandafillidi, National and Kapodistrian University of Athens, Athens, Greece
CROSS-COUPLING OF CHLORO(HETERO)ARENES WITH THIOLATES EMPLOYING A Ni-PRECATALYST
P. Gehrtz, Weizmann Institute, Rehovot, Israel
DEVELOPING NEW WAYS TO INTRODUCE THE BORON ATOM IN ORGANIC MOLECULES BY RING-OPENING REACTIONS
A. Menichetti, University of Pisa, Pisa, Italy
CATALYTICALLY ACTIVE PEPTIDES FOR CONJUGATE ADDITION REACTIONS
G. Vastakaite, ETH Zürich, Zürich, Switzerland
TANDEM INDIUM-MEDIATED REDUCTIVE REACTION/N-ANNULATION REACTION: SYNTHESIS OF BIS-PYRROLEARENE DERIVATIVES FROM ELECTRON DEFICIENT NITROANILINES
H. Lee, Dong-A University, Busan, Republic of Korea
SYNTHESIS OF UNPROTECTED, BICYCLIC AND SPIROCYCLIC β-AMINO ACIDS
H. Noda, Institute of Microbial Chemistry (BIKAKEN), Tokyo, Japan
LIGHT-RESPONSIVE LIGANDS CONTROLLING BIMETALLIC CATALYSTS FORMATION
H. El Said El Sayed , University of Twente, Enschede, The Netherlands
RADICAL CYCLIZATIONS OF A-OXY CARBON CENTERED RADICALS
E. Andre-Joyaux, University of Bern, Bern, Switzerland
REACTIVITY AND SYNTHETIC UTILITY OF α-BORYL CARBON CENTERED RADICALS: TWO OPPOSING REACTION MANIFOLDS
N. Tappin, University of Bern, Bern, Switzerland
DEVELOPMENT OF BICYCLO[1.1.0]BUTYL BORONATE COMPLEXES FOR THE DIASTEREOSELECTIVE SYNTHESIS OF CYCLOBUTANES
S. Bennett, University of Bristol, Bristol, UK
PHENYLGLYOXYLIC ACID AS THE CATALYST FOR PHOTOCHEMICAL TRANSFORMATIONS
C. Kokotos, National and Kapodistrian University of Athens, Athens, Greece
TRANSITION-METAL-MEDIATED RADICAL DEFORMYLATION OF ALDEHYDES USING VARIOUS AMINOXYL RADICALS
G. Schulz, Leibniz University Hannover, Hannover, Germany
DUAL LIGAND-ENABLED NONDIRECTED C-H CYANATION OF ARENES
A. Mondal, Max Planck Institute for Chemical Energy Conversion, Mülheim an der Ruhr, Germany
BORYLATION OF ALKYNES WITH CYCLODEXTRIN-ENCAPSULATED N-HETEROCYCLIC CARBENE COPPER COMPLEXES
S. Roland, Sorbonne Universités, Paris, France
HFIP SOLVENT ENABLES ALCOHOLS TO ACT AS ALKYLATING AGENTS IN STEREOSELECTIVE HETEROCYCLIZATION
Y. Zhu, University of Oxford, Oxford, UK
CONTROL OVER ENAMINE PYRAMIDALIZATION GIVES ACCESS TO N-HETEROCYCLIC SUBSTITUTED γ-NITROALDEHYDES
J. Möhler, ETH Zürich, Zürich, Switzerland
SWITCHABLE BASE METAL CATALYZED HYDROGEN BORROWING PROCESSES
N. Hofmann, University of Vienna, Vienna, Austria
DESIGN AND ASSESSMENT OF NOVEL POLYMERS BASED ON 5-DIHYDRAZINYL-1, 3,4-THIADIAZOLE AS INHIBITORS FOR STEEL PIPELINES CORROSION IN CO2-SATURATED OILFIELD
S. Al-Shihry, King Faisal University, Hufuf, Saudi Arabia
RHODIUM-CATALYZED REARRANGEMENT OF 2-FURYL TETHERED 1-TOSYL-1,2,3-TRIAZOLES
A.S. Makarov, Perm State University, Perm, Russia
Pd-CATALYZED TRIFLUOROMETHYLTHIOLATION OF ACRYLAMIDES AND AROMATIC AMIDES BY C-H BOND ACTIVATION
M.-Y. Chen, Normandie Université, Rouen, France
FORMAL SYNTHESIS OF PLATENCIN FROM O-VANILLIN BY INTERMOLECULAR AND INTRAMOLECULAR DIELS-ALDER STRATEGIES, RESPECTIVELY
D.-S. Hsu, National Chung Cheng University, Chiayi, Taiwan
ONE-POT MULTI-COMPONENT COUPLING-ADDITION SYNTHESIS OF HYDROXYPYRAZOLES, ALKOXYPYRAZOLES, AND β-AMINO ENOATES
J.S. Niedballa, Heinrich-Heine-University Düsseldorf, Düsseldorf, Germany
MONO- AND DISUBSTITUTED PSORALENS FOR INTERCALATION AND PHOTOADDITION INTO DNA
S.R. Geenen, Heinrich-Heine-University Düsseldorf, Düsseldorf, Germany
DIVERSITY-ORIENTED SYNTHESIS OF DIARYL SUBSTITUTED HERTEROCYCLES VIA SEQUENTIAL PALLADIUM CATALYSIS
L. Mayer, Heinrich-Heine-University Düsseldorf, Düsseldorf, Germany
REPLACING Cr(VI) WITH AN ENZYME: CLEAN OXIDATIONS
U. Hanefeld, Technische Universiteit Delft, Delft, The Netherlands
OPTIMIZED SYNTHESIS OF THE BACTERIAL MAGIC SPOT (p)ppGpp CHEMOSENSOR PyDPA
M. Minneci, Università degli Studi di Milano, Milan, Italy
C(sp3)–H ACETOXYLATION OF FREE CARBOXYLIC ACIDS
K.K. Ghosh, Westfälische Wilhelms-Universität Münster, Münster, Germany
TOWARDS THE TOTAL SYNTHESIS OF TIACUMICIN B: PREPARATION OF GLYCOSIDIC FRAGMENTS AND GLYCOSYLATION
S. Norsikian, ICSN CNRS-UPR 2301, Gif-sur-Yvette, France
ONE‐POT PREPARATION OF 1,2,3‐BENZOTRIAZIN‐4(3H)‐ONES AND ACETYLBENZOTRIAZOLES USING A KEY Cp*Co(III)‐CATALYZED C−H AMIDATION STEP
P. Chirila, Sheffield Hallam University, Sheffield, UK
STUDIES TOWARDS THE TOTAL SYNTHESIS OF DYSIHERBOL A
J. Erver, University of Cologne, Cologne, Germany
ENZYME-TRIGGERED CO-RELEASING MOLECULES (ET-CORMs) AS VERSATILE AND POWERFUL MEDICINAL AGENTS
B.M. Krause, University of Cologne, Cologne, Germany
STUDIES TOWARDS THE SYNTHESIS OF EURYSTEROL A
Ö. Taspinar, University of Cologne, Cologne, Germany
A NEW APPROACH TO PREPARE α-FLUORINATED β-AMINO ACIDS, BEARING A TETRASUBSTITUTED STEREOGENIC CENTER
I. Eder, Johannes Kepler University Linz, Linz, Austria
STEREOSELECTIVE SYNTHESIS OF SATURATED NITROGEN HETEROCYCLES VIA HYDROGEN BORROWING CATALYSIS
A. Chamberlain, University of Oxford, Oxford, UK
CARBOMETALLATION OF CYCLOPROPENYLSILANES
Y. Cohen, Israel Institute of Technology, Haifa, Israel
REMOTE FUNCTIONALIZATION OF STEREODEFINED SUBSTITUTED CYCLOPROPANES
A. Cohen, Israel Institute of Technology, Haifa, Israel
MOLECULAR ADSORBATES SWITCH ON HETEROGENEOUS CATALYSIS: INDUCTION OF REACTIVITY BY N-HETEROCYCLIC CARBENES
M. Das, Westfälische Wilhelms-Universität Münster, Münster, Germany
CYCLOPROPANATION OF ALIPHATIC ESTERS AND ALCOHOLS EXTENDED TO ONE-STEP CATALYTIC LINEAR SULFONE
T. Vojkovsky, Okinawa Institute of Science and Technology Graduate University, Onna, Japan
SYNTHESIS AND APPLICATIONS OF CHIRAL QUATERNARY AMMONIUM SALT HYDROGEN BOND DONOR CATALYSTS
V. Haider, Johannes Kepler University Linz, Linz, Austria
HIGHLY ENANTIOSELECTIVE PHASE-TRANSFER CATALYZED ADDITION OF ISOXAZOLIDIN-5-ONES TO MBH CARBONATES AND PARA QUINONE METHIDES: ACCESS TO FUNCTIONALIZED β2,2-AMINO ACIDS
A. Eitzinger, Johannes Kepler University Linz, Linz, Austria
UMPOLUNG REACTIONS OF IMINES FOR THE SYNTHESES OF α-TRIFLUOROMETHYLATED AMINO ACIDS
M. Winter, Johannes Kepler University Linz, Linz, Austria
ACCEPTOR METAL-DIRECTED SUPRAMOLECULAR TOPOLOGIES
D.H. Kim, University of Ulsan, Ulsan, Republic of Korea
SYNTHESIS AND CHEMICAL MODIFICATIONS OF PEPTIDE CONJUGATES:INVESTIGATING PEPTIDE-PROTEIN INTERACTIONS
A. Balliu , Stockholm University, Stockholm, Sweden
SYNTHESIS OF MACROCYCLIC COMPOUNDS VIA CONSECUTIVE SONOGASHIRA-UGI-SONOGASHIRA REACTIONS
M. Glavaš, Ruđer Bošković Institute, Zagreb, Croatia
A MILD AND DIRECT SITE-SELECTIVE sp2 C-H SILYLATION OF (POLY)AZINES
Y. Gu, The Barcelona Institute of Science and Technology, Tarragona, Spain
CONTROL OVER SURFACE WETTABILITY BY SURFACE-IMMOBILISED MOLECULAR MOTORS
C.L.F. van Beek, University of Groningen, Groningen, The Netherlands
MAKING THE UNDRUGGABLE DRUGGABLE: SYNTHETIC PROLIN-DERIVED MODULES (ProMs) AS BUILDING BLOCKS FOR RATIONAL AND LIBRARY-BASED DRUG DEVELOPMENT
S. Chiha, University of Cologne, Cologne, Germany
A "TOP DOWN" APPROACH TO THE SYNTHESIS OF COMPLEX, DIVERSE LEAD-LIKE SCAFFOLDS
E. Okolo, University of Leeds, Leeds, United Kingdom
NOVEL APPROACHES TO 2-AMINOBENZOXAZOLES
V. Šlachtová, Palacky University, Olomouc, Czech Republic
PHOTOCHROMIC PEPTIDES FOR LIGHT-TRIGGERED DRUG DELIVERY AND BEYOND
S. Kirchner, Karlsruhe Institute of Technology, Karlsruhe, Germany
CARBOXYLATE CATALYSED ISOMERISATION OF UNSATURATED NAC-THIOESTERS
S. Riuttamäki, University of Jyväskyla, Jyväskyla, Finland
SYNTHESIS AND CHARACTERIZATION OF SERS-ACTIVE HETEROAROMATIC MOLECULES
F. Fontana, University of Bergamo, Bergamo, Italy
LATE-STAGE FUNCTIONALIZATION OF PEPTIDES AND CYCLOPEPTIDES USING ORGANOZINC REAGENTS
M. Leroux, Ludwig-Maximilians University, Munich, Germany
NOVEL PATHWAY TOWARDS STANNYLATED GLUCALS
A. Klaiber, University of Tübingen, Tübingen, Germany
SYNTHETIC PATHWAYS TOWARDS CARBOHYDRATE-SUBSTITUTED ALPHA-DIKETONES
A. Daikeler, University of Tübingen, Tübingen, Germany
CARBOHYDRATE DERIVED LIGANDS FOR CATALYTIC STEREOSELECTIVE CARBENOID CYCLOPROPANATION REACTIONS
F. Preusch, University of Tübingen, Tübingen, Germany
THE SYNTHESIS OF CARBON BRIDGED C-DISACCHARIDES VIA LITHIATED GLYCALS
J. Kessler, University of Tübingen, Tübingen, Germany
SYNTHESIS OF NEW GLYCOPEPTIDES
L. Srsan, University of Tübingen, Tübingen, Germany
THE SYNTHESIS OF DODECO-6,7-DIULOSES
M. Bayer, University of Tübingen, Tübingen, Germany
GLYCOCONJUGATED AB3-SECO-PORPHYRAZINES AS POTENTIAL PHOTOSENSITIZERS IN PHOTODYNAMIC THERAPY
Th. Klein, University of Tübingen, Tübingen, Germany
SYNTHESIS OF NOVEL AZA-BODIPY DERIVATES FOR PHOTODYNAMIC THERAPY
T. Zweiböhmer, University of Tübingen, Tübingen, Germany
SYNTHESIS OF NEW STERICAL DEMANDING CHIRAL AMINES
J. Dürner, Technical University Munich, Garching, Germany
SURPRISINGLY SIMPLE CATALYTIC ACCESS TO STEREODEFINED FULLY-SUBSTITUTED ALDEHYDE ENOLATES
I. Massad, Israel Institute of Technology, Haifa, Israel
AN ELECTROCHEMICAL APPROACH TO RADICAL TRIFLUOROMETHYLATIONS AND OXYTRIFLUOROMETHYLATIONS
W. Jud, University of Graz, Graz, Austria
COPPER CATALYZED ASYMMETRIC FORMATION OF ENANTIOENRICHED β-CF3 ESTER & NITRILE DERIVATIVES
P. Poutrel, Normandie Université, Rouen, France
N-HETEROCYLIC CARBENE CONTROLLED DIVERGENT DEHOMOLOGATION OF ALDOSES
M. Draskovits, TU Wien, Vienna, Austria
COPPER CATALYSED AND ADDITIVE FREE DECARBOXYLATIVE TRIFLUOROMETHYLATION OF (HETERO)AROMATIC IODIDES
M. Johansen, Aarhus University, Aarhus, Denmark
COPPER-CATALYZED BORYLATION OF OLEFINS: A QUEST FOR REACTIVITY AND SELECTIVITY
D. Fiorito, University of Geneva, Geneva, Switzerland
ENANTIOSELECTIVE NICKEL-CATALYZED AMINATION OF 2-SUBSTITUTED 1,3-DIENES
G. Tran, University of Geneva, Geneva, Switzerland
SUPRAMOLECULARLY REGULATED COPPER-BISOXAZOLINE CATALYSTS FOR THE EFFICIENT INSERTION OF CARBENOID SPECIES INTO HYDROXYL BONDS
E. Iniesta , The Barcelona Institute of Science and Technology, Tarragona, Spain
TOWARDS THE TOTAL SYNTHESIS OF VIOPROLIDES A-D
H. Grab, Technical University Munich, Garching, Germany
PHOTOCHEMICAL REACTION CASCADE FROM O-PENT-4-ENYL-SUBSTITUTED SALICYLATES TO COMPLEX MULTIFUNCTIONAL SCAFFOLDS
A. Zech, Technical University Munich, Garching, Germany
ELECTROCATALYTIC IODOPERFLUOROALKYLATION OF UNSATURATED HYDROCARBONS
M. Sommer, Heinrich-Heine-University Düsseldorf, Düsseldorf, Germany
ALKOXYDIPHENYLPHOSPHINITES AS CARBOCATION SYNTHONS
L. Ochmann, Justus Liebig University Giessen, Giessen, Germany
LEWIS-ACID CATALYZED PHOTOREARRANGEMENT OF 2,4-CYCLOHEXADIENONES
M. Leverenz, Technical University Munich, Garching, Germany
TOWARDS THE TOTAL SYNTHESIS OF (-)-PULVOMYCIN
S. Wienhold, Technical University Munich, Garching, Germany
METABOLISM MIMICRY: AN ELECTROSYNTHETIC METHOD FOR THE SELECTIVE DEETHYLATION OF TERTIARY BENZAMIDES
M.K. Bal, Manchester Metropolitan University, Manchester, United Kingdom
DEVELOPING NOVEL PET TRACERS FOR HYPOXIA
F. Angelucci, University of Bergen, Bergen, Norway
DRUG REPURPOSING: SULFASALAZINE AS A NEW ANTICANCER TREATMENT. STUDY OF TUMOUR DRUG DISTRIBUTION THROUGH PET AND MRI IMAGING
D. Cirillo, University of Bergen, Bergen, Norway
MOLECULAR Co-CORROLE COMPLEX FOR THE HETEROGENEOUS ELECTROCATALYTIC REDUCTION OF CARBON DIOXIDE ON CARBON FIBER ELECTRODES
S. Gonglach, Johannes Kepler University Linz, Linz, Austria
INCREASING THE π-ELECTRON CONJUGATION OF CORROLES VIA SONOGASHIRA-CROSS-COUPLING
M. Haas, Johannes Kepler University Linz, Linz, Austria
ERINE 2425.46 AND ALANINE 2225.46 AS DETERMINANTS OF 5-HT2A/2C SELECTIVITY
T. Chávez, University of Chile, Santiago, Chile
SYNTHETIC KETOREDUCTASE MIMICS
T. Metsänen, University of Jyväskyla, Jyväskyla, Finland
In/Ag-CATALYZED CONSTRUCTION OF N-ARYLPYRAZOLES VIA REGIOSELECTIVE [2+2+1]-OXIDATIVE N-ANNULATION: TWO IS BETTER THAN ONE
R.S. Thombal, Yeungnam University, Gyeongsan, Republic of Korea
METAL- FREE BASE MEDIATED TANDEM BENZANNULATION OF N-TOSYLHYDRAZONES WITH 3 FORMYLCHROMONES: A GENERAL ROUTE TO DIVERSE AND POLYFUNCTIONALIZED XANTHONES
R. Shrestha, Yeungnam University, Gyeongsan, Republic of Korea
Cγ-SUBSTITUENTS AS TOOLS TO INFLUENCE THE REACTIVITY AND STEREOSELECTIVITY OF PROLINE BASED CATALYSTS
M. Schnurr, ETH Zürich, Zürich, Switzerland
CARBON DIOXIDE-CATALYZED STEREOSELECTIVE CYANATION OF COUMARINS
T. Roy, University of Copenhagen, Copenhagen, Denmark
SYNTHESIS OF THE DIARYLACETYLENES BEARING ELECTRON WITHDRAWING GROUP VIA THE SMILES REARRANGEMENT
R. Bujok, Polish Academy of Science, Warsaw, Poland
FLUOROPHOBIC EFFECT LEADS TO NOVEL LIQUID CRYSTALLINE DONOR ACCEPTOR DYES
F. Schulz, University of Stuttgart, Stuttgart, Germany
STEREOCONTROLLED DEBENZYLATING CYCLOETHERIFICATION DEPENDED ON SUBSTRATE REACTIVITY
K. Tiara, Polish Academy of Science, Warsaw, Poland
FIRST SYNTHESIS OF CRYPTANDS WITH SUCROSE SCAFFOLD
P. Sokołowska, Polish Academy of Science, Warsaw, Poland
SYNTHESIS AND BIOLOGICAL PROFILING OF MEPHEDRONE METABOLITES
D. Cintulova, TU Wien, Vienna, Austria
SYNTHESIS OF THE AB RING SYSTEM OF CLIFEDNAMIDE
M. Sinast, University of Stuttgart, Stuttgart, Germany
COMPARISON OF TWO SYNTHETIC STRATEGIES TOWARDS 1-ACYL-2-VINYLCYCLOPROPANES
M. Holzwarth, University of Stuttgart, Stuttgart, Germany
UNPRECEDENTED MULTICOMPONENT ORGANOCATALYTIC SYNTHESIS OF PROPARGYLIC ESTERS VIA CO2 ACTIVATION
M. Pauze, University of the Basque Country, Donostia/San Sebastian, Spain
NOVEL CHK1 INHIBITOR MU380 EXHIBITS SIGNIFICANT SINGLE-AGENT ACTIVITY IN TP53-MUTATED CHRONIC LYMPHOCYTIC LEUKEMIA CELLS
P. Khirsariya, Masaryk University, Brno, Czech Republic
VICARIOUS NUCLEOPHILIC CHLOROMETHYLATION OF NITROAROMATICS
V. Khutorianskyi, Academy of Science of the Czech Republic, Prague, Czech Republic
A PRELIMINARY STUDY ON THE REGIOSELECTIVE C-H ARYLATION OF IMIDAZO[2,1-b]THIAZOLE
M. Lessi, Universita di Pisa, Pisa, Italy
RADICAL FLUOROALKYLATION OF NITROGEN HETEROCYCLES AND AROMATIC AMINO ACID RESIDUES IN PEPTIDES AND PROTEINS
K. Rahimidashaghoul, Academy of Science of the Czech Republic, Prague, Czech Republic
DONOR–ACCEPTOR CYCLOPROPANES: A REACTIVITY STUDY
A. Kreft, TU Braunschweig, Braunschweig, Germany
IRON-CATALYZED CYCLOPROPANATION OF 1,3-ENYNES UNDER THERMAL OR PHOTOCHEMICAL CONDITIONS
M.-I. Picher, University of Stuttgart, Stuttgart, Germany
CYCLIZATION OF 5-(1H-INDOL-3-YL)-3-OXOPENTANOIC ACID ESTERS AND AMIDES PROMOTED WITH TRANSITION METAL TRIFLATES
M. Szewczyk, Gdansk University of Technology, Gdansk, Poland
Zn(II)-CATALYZED [3+2] AND [4+2] ANNULATION OF INDOLES WITH AZOALKENES: DIVERGENT SYNTHESIS OF POLYCYCLIC INDOLINES
C. Ciccolini, University of Urbino "Carlo Bo", Urbino, Italy
PHOTOCATALYTIC TRANSFORMATIONS OF ALKENES: STUDIES ON PHOTOREDUCTION AND E→Z ISOMERIZATION
J. Miyatake Ondozabal, University of London, London, United Kingdom
SYNTHESIS AND CHARACTERIZATION OF NON-PLANAR TETRAAZAPEROPYRENES (TAPPS) VIA BAY-SUBSTITUTION
B. Günther, Heidelberg University, Heidelberg, Germany
AN ENTRY TO ENANTIOENRICHED ALLYLAMINES VIA PHOTOCHEMICAL CROSS-COUPLING AND ICHIKAWA REARRANGEMENT
M. Garbacz, Polish Academy of Science, Warsaw, Poland
ALKENE HYDROSILYLATION CATALYZED BY EASILY ASSEMBLED Ni(II)-CARBOXYLATE MOFs
Z. Zhang, Ecole Polytechnique Federale de Lausanne (EPFL), Lausanne, Switzerland
CHROMOPHORE ACTIVATION AT ITS BEST - INFLUENCING THE SELECTIVITY OF PHOTOREACTIONS BY ADDITION OF LEWIS ACIDS
S. Stegbauer, Technical University Munich, Garching, Germany
HIGHLY ENANTIOSELECTIVE CHROMIUM(II) PINCER CATALYZED HYDROSILYLATION OF KETONES
Ch. Schiwek, Technical University of Munich, Munich, Germany
REACTION INTERMEDIATES IN PALLADIUM-CATALYZED CARBONYLATION OF OLEFINS
M. Anania, Charles University, Prague, Czech Republic
THE SYNTHESIS OF AN ARTIFICIAL, BACKBONE MODIFIED ENTEROBACTIN ANALOGUE
R. Zscherp, Technical University of Braunschweig, Braunschweig, Germany
DIVERGENT ACCESS TO HISTONE DEACETYLASE INHIBITORY CYCLOPEPTIDES VIA LATE-STAGE CYCLOPROPANE RING CLEAVAGE STRATEGY. SHORT TOTAL SYNTHESIS OF CHLAMYDOCIN
G.Z. Elek, Tallinn University of Technology, Tallinn, Estonia
A SHORT SYNTHETIC APPROACH TO A LIBRARY OF NON NATURAL PPAP DERIVATIVES WITH ANTIMICROBIAL PROPERTIES AND INSIGHTS INTO THEIR ANTIBIOTIC MECHANISM
F. Kraus, University of Stuttgart, Stuttgart, Germany
VISIBLE-LIGHT-MEDIATED α-OXYGENATION OF 3-(N,N-DIMETHYLAMINOMETHYL)-INDOLES TO ALDEHYDES
F. Stanek, Polish Academy of Science, Warsaw, Poland
EXPLOITING ORGANOSULFUR COMPOUNDS IN DONOR-ACCEPTOR CYCLOPROPANE CHEMISTRY
A.U. Augustin, TU Braunschweig, Braunschweig, Germany
N-FLUOROALKYL-1,2,3-TRIAZOLES: EASILY AVAILABLE COMPOUNDS WITH HIGH SYNTHETIC POTENTIAL
A. Markos, Academy of Science of the Czech Republic, Prague, Czech Republic
DIVERGENT 1,3-DIFUNCTIONALIZATION OF AMINOCYCLOPROPANES
M.-M. Wang, Ecole Polytechnique Federale de Lausanne (EPFL), Lausanne, Switzerland
SIGMATROPIC REARRANGEMENT OF IMINIUM SALTS EXEMPLIFIED ON NORADAMANTANE DERIVATIVES
B. Zonker, Justus Liebig University Giessen, Giessen, Germany
IRON-CATALYSED HYDROBORATION OF UNSATURATED C-C BONDS: BORON-SOURCE CONTROLLED SELECTIVITY
F. Rami, University of Stuttgart, Stuttgart, Germany
DOUBLE ELECTROPHILIC ACTIVATION OF YNAMIDES: A STRAIGHTFORWARD ENTRY TO α-HALO-CARBOXYL DERIVATIVES
P. Thilmany, Université libre de Bruxelles, Bruxelles, Belgium
TOWARDS THE TOTAL SYNTHESIS OF PECTENOTOXIN-4
T. Kwok, University of Oxford, Oxford, UK
SYNTHESIS OF A NOVEL CYCLIC PEPTIDE LIBRARY ENABLED BY C-H FUNCTIONALIZATIONS AND THE DNA-ENCODED LIBRARY TECHNOLOGY
M. Pourghasemi Lati, Stockholm University, Stockholm, Sweden
PHOTOREDOX-MEDIATED RADICAL DIFUNCTIONALIZATION OF CYCLOPROPENES
B. Muriel, Ecole Polytechnique Federale de Lausanne (EPFL), Lausanne, Switzerland
FACILE SYNTHESIS OF DIVERSE BENZOPYRAN DERIVATIVES VIA GOLD-CATALYZED CYCLIZATION AND GENERATION OF ARYNES
Y. Nakamura, Tokyo Medical and Dental University (TMDU), Tokyo, Japan
TOTAL SYNTHESIS OF PALIURINE E: A HIGHLY CONVERGENT "BLOCK" APPROACH
D. Dewez, Université libre de Bruxelles, Bruxelles, Belgium
CHEMOSELECTIVE COPPER(I)-CATALYZED CONJUGATE REDUCTIONS OF ENOATES USING H2
B.M. Zimmermann, Technische Universität Berlin, Berlin, Germany
USING H2 AS A HYDRIDE SOURCE - A CHEMO- AND REGIOSELECTIVE REDUCTIVE COUPLING REACTION/ALLYLIC REDUCTION
L.T. Brechmann, Technische Universität Berlin, Berlin, Germany
Ni-CATALYZED E-SELECTIVE ALKYNE SEMIHYDROGENATIONS
B. Kaewmee, Technische Universität Berlin, Berlin, Germany
A SHORT TOTAL SYNTHESIS OF NATURAL CARBASUGAR
S. Holmstedt, Tampere University, Tampere, Finland
MULTISTEP CONTINUOUS FLOW SYNTHESIS OF THE CHIRAL KEY INTERMEDIATE OF PAROXETINE
S.B. Ötvös, University of Graz, Graz, Austria
NICKEL CATALYZED HYDROXYCARBONYLATION OF ACETYLENE TO ACRYLIC ACID
H.S. Choi, Korea Research Institute of Chemical Technology, Daejeon, Republic of Korea
CAGING AND CONTROLLED RELEASE OF AN ANTIBACTERIAL DRUG BY CELL SURFACE FUNCTIONALIZATION
I. Shchelik , University of Zurich, Zurich, Switzerland
ENANTIOSELECTIVE SYNTHESIS OF CHROMANONES WITH QUARTENARY STEREOGENIC CENTER VIA NHC ORGANOCATALYSIS
K. Dzieszkowski, Nicolaus Copernicus University, Toruń, Poland
KINETIC QUANTIFICATION OF ALDOSE OPEN-CHAIN CONTENT
H. Kalaus, TU Wien, Vienna, Austria
CONDUCTIVITY STUDIES OF DIARLYETHYLENE-MODIFIED DNA VIA SCANNING TUNNELING MICROSCOPY
M. Schupp, Karlsruhe Institute of Technology, Karlsruhe, Germany
ENANTIOSELECTIVE C-H ACTIVATION WITH Rh(I)JasCp COMPLEXES
S. Shaaban, Max-Planck-Institute for Molecular Physiology, Dortmund, Germany
SYNTHESIS AND ANTICANCER ACTIVITY OF 2-(1,3,5-TRIAZIN-2-YLMETHYLTHIO)-N-(IMIDAZOLIDIN-2-YLIDENE)-5-METHYL BENZENESULFONAMIDE DERIVATIVES
Ł. Tomorowicz, Medical University of Gdańsk, Gdańsk, Poland
RHODIUM-CATALYZED REGIOSELECTIVE ACTIVATION OF STERICALLY HINDERED C-C BOND OF BIPHENYLENE
H. Takano, Waseda University, Tokyo, Japan
SYNTHESIS OF FUNCTIONALIZED MOLECULAR TRIPODS FOR SURFACE APPLICATIONS
N. Balzer, Karlsruhe Institute of Technology, Karlsruhe, Germany
AMORPHOUS PURINE-AZOLE CONJUGATES AND THEIR PHOTOPHYSICAL PROPERTIES
A. Sebris, Riga Technical University, Riga, Latvia
CATIONIC 1,2-SILYL SHIFT IN PROPARGYL SILANES
M. Puriņš, Riga Technical University, Riga, Latvia
DEVELOPMENT OF A NOVEL LIGATION STRATEGY FOR SYNTHESIS OF THERAPEUTIC GLYCOPEPTIDES
D. Lynch, Trinity College Dublin, Dublin, Ireland
PHOTOREDOX MEDIATED SYNTHESIS OF SULFINATE ESTERS FROM TOSYLHYDRAZONE SUBSTRATES
J. Slater, Sheffield Hallam University, Sheffield, UK
SYNTHESIS OF A POTENTIAL COMPOUND BASED ON A DIAMINODIPHENYLBUTADIENE TO REPAIR DNA-LESIONS
G.M. Rodriguez-Muñiz, Universitat Politécnica de València, València, Spain
DEVELOPMENT OF NOVEL THIOL-ENE MEDIATED PEPTIDE LIGATION STRATEGIES
J. McLean, Trinity College Dublin, Dublin, Ireland
STUDIES TOWARD THE TOTAL SYNTHESIS OF NAHUOIC ACID A
B. Stoessel, ETH Zürich, Zürich, Switzerland
SYNTHESIS OF VERSATILE BICYCLOPENTANE BUILDING BLOCKS FROM [1.1.1]PROPELLANE
G.L. Tolnai, Eotvos Lorand University, Budapest, Hungary
COPPER CATALYZED RING OPENING REACTIONS OF [1.1.1]PROPELLANE
D. Lasányi, Eotvos Lorand University, Budapest, Hungary
CROWN ETHER-BASED MESOGENS WITH BRANCHED ALKYL CHAINS
P. Seubert, University of Stuttgart, Stuttgart, Germany
PHOTOREDOX-CATALYZED ALKYLATION OF HETEROAROMATIC BASES USING ETHYL ACETATE AS ALKYLATING AGENT
N. Győrfi, Servier Research Institute of Medicinal Chemistry, Budapest, Hungary
STEREOSELECTIVE MODIFICATION OF "α-HYDROXY ACID PEPTIDES" BY PALLADIUM CATALYZED ALLYLIC ALKYLATION
A. Horn, Saarland University, Saarbrücken, Germany
COLOR TUNING OF ELECTROCHROMIC HETEROPHENOQUINONES
S. Intorp, Ruprecht-Karl-University Heidelberg, Heidelberg, Germany
ELECTRON-HOLE CATALYZED ORTHO-HYDROARYLATION
B. Özkaya, RWTH Aachen University, Aachen, Germany
A CLICK-CHEMISTRY LINKED 2’3’-cGAMP ANALOGUE
C. Dialer, Ludwig-Maximilians University, Munich, Germany
SYNTHESIS OF 1,2-DIAZETIDIN-3-ONES VIA THE UGI REACTION COMPRISING α-HYDRAZINO ACIDS
I. Jeric, Ruđer Bošković Institute, Zagreb, Croatia
DNA FROM AN ELECTRICAL POINT OF VIEW - POTENTIAL BUILDING BLOCKS FOR MOLECULAR ELECTRONICS
Ch. Bickmann, Karlsruhe Institute of Technology, Karlsruhe, Germany
SHORT PEPTIDES WITH PHOTOCATALYTIC ACTIVITY FOR THE NUCLEOPHILIC ADDITION OF METHANOL TO STYRENE DERIVATIVES
D. Sack, Karlsruhe Institute of Technology, Karlsruhe, Germany
PHENOTHIAZINIMIDES: ATOM-EFFICIENT ELECTROPHILIC AMINATION REAGENTS
Ch. Bub, RWTH Aachen University, Aachen, Germany
LATE-STAGE INDOLE SYNTHESIS ENABLES THE TOTAL SYNTHESIS OF TRYPTOPHAN CONTAINING PEPTIDES
L. Junk, Saarland University, Saarbrücken, Germany
SYNTHESIS OF AMORPHOUS FLUORESCENT PURINE HYBRIDS CONTAINING FIVE-MEMBERED HETEROCYCLES
Z. Kapilinskis, Riga Technical University, Riga, Latvia
ONE-STEP SYNTHESIS OF SUBSTITUTED 2-OXAZOLIDINONES VIA BASE-CATALYZED CO2-FIXATION AND AZA-MICHAEL ADDITION
J. Mannisto, University of Helsinki, Helsinki, Finland
A STEREOFLEXIBLE ACCESS TO 2-ALKENYLATED INDOLES
T. Hergert, Budapest University of Technology and Economics, Budapest, Hungary
NOVEL ADDRESSABLE CHOLESTEROL ANALOGUES FOR LIVE IMGAGING OF CELLULAR MEMBRANES
T. Wegner, Westfälische Wilhelms-Universität Münster, Münster, Germany
COMPUTATIONAL DESIGN OF NOVEL BICYCLO[2.2.2]OCTANE BASED PROTON SPONGES
Z. Glasovac, Ruđer Bošković Institute, Zagreb, Croatia
RHODIUM CATALYZED CYCLOPROPANATION WITH α-ALKYL-α-DIAZO ESTERS
Ch. Zippel, Karlsruhe Institute of Technology, Karlsruhe, Germany
NEW MODIFICATIONS OF AN OLD SCAFFOLD: PYRAZOLOQUINOLINONE DERIVATIVES AND ANALOGUES AS ACTIVE COMPOUNDS ON GABAA RECEPTORS
M. Iorio, TU Wien, Vienna, Austria
NOVEL Mg-BASED APPROACH FOR THE REGIOSELECTIVE FUNCTIONALIZATION OF PURINE DERIVATIVES
S. Gazzola, University of Insubria, Como, Italy
DIALKYLATION OF 1,3-DIENES BY DUAL PHOTOREDOX AND CHROMIUM CATALYSIS
H.-M. Huang, Westfälische Wilhelms-Universität Münster, Münster, Germany
ASYMMETRIC LACTONE SYNTHESIS BY REDUCTIVE OLEFIN ACTIVATION AND CO2-FIXATION
A. Sahari, University of Helsinki, Helsinki, Finland
NOVEL β-AMINO ACID DERIVED ASYMMETRIC ORGANOCATALYSTS TOWARDS 3,3-DISUBSTITUTED-2-OXINDOLES’
M. Gavendova, Waterford Institute of Technology, Waterford, Ireland
Cu(II)-CATALYZED CROSS-DEHYDROGENATIVE ORTHO-AMINOMETHYLATION OF PHENOLS
C. Yu, RWTH Aachen University, Aachen, Germany
DUAL PHOTOREDOX CATALYSED sp2-sp3 CROSS-ELECTROPHILE COUPLING IN A SELF-DESIGNED AND 3D PRINTED PHOTOREACTOR
F. Schiel, Boehringer Ingelheim RCV GmbH & Co KG, Vienna, Austria
OXIDATIVE PHENOL COUPLING IN NATURAL PRODUCT SYNTHESIS
J. Greb, Heinrich-Heine-University Düsseldorf, Jülich, Germany
STEREOSELECTIVE ACID-CATALYZED C(sp3)-C(sp3) BOND FORMATION IN THE INTRAMOLECULAR SYNTHESIS OF cis-1,2-DIARYL CYCLOPROPANES
I. Madarász, AVICOR Ltd., Szeged, Hungary
SYNTHESIS OF DOUBLE-CLICK AZOBENZENES FOR AN EASY FUNCTIONALIZATION OF BIOMOLECULES
R. Conceicao, TU Wien, Vienna, Austria
DIASTEREODIVERGENT SYNTHESIS OF ENANTIOENRICHED α,β-DISUBSTITUTED γ-BUTYROLACTONES VIA COOPERATIVE CATALYSIS
E. Serrano, Westfälische Wilhelms-Universität Münster, Münster, Germany
2,2-DIMETHYL-2H-PYRANS: DIENES FOR DOMINO DIELS-ALDER / RETRO DIELS-ALDER REACTIONS IN THE SYNTHESIS OF POLYSUBSTITUTED 2-NAPHTOATES
A. Díaz, Instituto de Productos Naturales y Agrobiología, Tenerife, Spain
CENTROSYMMETRIC APPROACH TOWARDS THE SYNTHESIS OF FUSED POLYCYCLIC ETHER NATURAL PRODUCTS
J. Elwood, University of Glasgow, Glasgow, United Kingdom
DIASTEREOSELECTIVE PALLADIUM-CATALYZED C–H ARYLATION OF FERROCENYLMETANEAMINES WITH ARYLBORONIC ACIDS AND PINACOL ESTERS
B. Mudráková, Comenius University Bratislava, Bratislava, Slovakia
STEREOSELECTIVE MICHAEL ADDITION OF ALDEHYDES TO HETEROCYCLIC NITROALKENES CATALYZED BY HYBRID PEPTIDE-THIOUREA CATALYSTS
P. Čmelová, Comenius University Bratislava, Bratislava, Slovakia
SYNTHESIS AND OPTIMIZATION OF 10H-PHENOTHIAZINE ANALOGUES FOR THE INHIBITION OF AUTOPHAGY
E. Alme, University of Bergen, Bergen, Norway
ONE-STEP SYNTHESIS OF ISOINDOLO[2,1-a]INDOL-6-ONES VIA TANDEM Pd-CATALYZED AMINOCARBONYLATION AND C-H ACTIVATION REACTION
T. Čarný, Slovak University of Technology, Bratislava, Slovakia
FIRST TOTAL SYNTHESIS OF VARIOXIRANOL A
M. Stiblarikova, Slovak University of Technology, Bratislava, Slovakia
FACILE ACCESS TO NITROARENES AND NITROHETEROARENES USING N-NITROSACCHARIN: AN ELECTROPHILIC NITRATING REAGENT
R. Calvo, Swiss Federal Institute of Technology, Zürich, Switzerland
ENANTIOSELECTIVE SYNTHESIS OF N-BENZYLIC HETEROCYCLES: A NICKEL- AND PHOTOREDOX-DUAL CATALYSIS APPROACH
C. Pezzetta, Dr. Reddy’s Laboratories Ltd., Cambridge, UK
SYNTHESIS AND STRUCTURE OF REGIOREGULAR POLY(1,4-POLY-ARYLENE)
Y. Shibuya, Kobe University, Kobe, Japan
SYNTHETIC STUDIES ON LAMELLARINS
K. Morii, Kobe University, Kobe, Japan
SYNTHESIS OF DIVERSE BENZOTHIOPHENES VIA REACTION OF ARYNES WITH ALKYNYL SULFIDES
T. Matsuzawa, Tokyo Medical and Dental University (TMDU), Tokyo, Japan
GENERATION AND UTILIZATION OF UNSTABLE CARBENOID INTERMEDIATES USING CONTINUOUS FLOW TECHNOLOGY
T. von Keutz, University of Graz, Graz, Austria
SYNTHESIS OF BENZOFURANYLINDOLINONES ANDSPIRONAPHTHOQUINONESBY REACTION OF 3-SUBSTITUTED PHTHALIDES AND OXINDOLE DERIVED NITRO-OLEFINS
S. Alati, Indian Institute of Technology Bombay, Mumbai, India
SYNTHESIS OF FUNCTIONALIZED OLEFINS VIA BASE MEDIATED 1,6-ADDITION OF DIAZO COMPOUNDS AND THEIR ACTIVE METHYLENE PRECURSORS TO p-QUINONE METHIDES
S. Pati, Indian Institute of Technology Bombay, Mumbai, India
IMPROVED SYNTHESIS OF DEUTERIUM LABELED ATYPICAL BILE ACID METABOLITES AS ANALYTICAL STANDARDS FOR BILE ACID DISORDER DIAGNOSIS
A. Sferrazza, IRBM SpA, Rome, Italy
SECONDARY STRUCTURAL MOTIFS IN DISUBSTITUTED FERROCENE AMIDES
S. Opačak, The Ruđer Bošković Institute, Zagreb, Croatia
NOVEL FUNCTIONALITYS OF ADOMET ANALOGS FOR NUCLEIC ACIDS LABELING
V. Masevicius, Vilnius University, Vilnius, Lithuania
A DFT STUDY OF REGIOSELECTIVITY IN DIELS-ALDER CYCLOADDITION OF E-BENZILIDENEGUANIDINE WITH 4,5-, 5,6- AND 6,7- INDOLYNES
I. Antol, The Ruđer Bošković Institute, Zagreb, Croatia
CARBAMOYLATED ENAMINONES AS VERSATILE BUILDING BLOCKS FOR THE SYNTHESIS OF AZAHETEROCYCLES
D. Obydennov, The Ural Federal University, Ekaterinburg, Russia
CONTINUOUS FLOW APPROACH FOR THE SYNTHESIS OF MAYTANSINOL, AS ADC-BASED THERAPY CYTOTOXIC AGENT
S. Princiotto, Università degli Studi di Siena, Siena, Italy
ENANTIOSELECTIVE BENZOIN REACTION CATALYZED BY N-HETEROCYCLIC CARBENE BORONIC ESTERS (NHC-BE)
V. Dhayalan, University of the Negev, Beer-Sheva, Israel
A BROADLY APPLICABLE AND STRAIGHTFORWARD ENTRY TO SELECTIVELY DEUTERATED AMINES
M. Lahboubi, Université libre de Bruxelles, Bruxelles, Belgium
BACTACS: A POTENTIAL STRATEGY FOR THE SELECTIVE DEGRADATION OF PROTEINS WITHIN PROKARYOTES
G. Brodie, University of Glasgow, Glasgow, United Kingdom
A UNIFIED APPROACH TO THE CHEMOSELECTIVE ALPHA-FUNCTIONALIZATION OF AMIDES
M. Lemmerer, University of Vienna, Vienna, Austria
A CHIMERA MODEL OF RelSeq PRE-CATALYTIC STATE
M. Civera, Università degli Studi di Milano, Milan, Italy
IBX/NIS INDUCED OXIDATIVE INTRAMOLECULAR ANNULATION
Z. Makra, AVIDIN Ltd., Szeged, Hungary
ACTIVATED THIOCYANATES - THE CYANOSULFENYLATION OF INTERNAL ALKYNES
M. Bürger, Technical University of Braunschweig, Braunschweig, Germany
COPPER CATALYZED 1,4-BROOK REARRANGEMENT OF α,β-UNSATURATED ACYLSILANE
G. Marghem, Université Catholique de Louvain (UCL), Louvain-la-Neuve, Belgium
HIGHLY ENANTIOSELECTIVE IRON-CATALYZED REDUCTION OF FUNCTIONALIZED KETONES AND NON-PRIVILEGED IMINES
C. Blasius, Ruprecht-Karl-University Heidelberg, Heidelberg, Germany
TRIFUNCTIONAL SELF-IMMOLATIVE SPACERS LINKED TO AMIDES: A NEW OPPORTUNITY FOR BIOCONJUGATION
A. Petrini, Università degli Studi di Siena, Siena, Italy
FORMAL SEMISYNTHESIS OF DEMETHYLGORGOSTEROL USING AN ENANTIOSELECTIVE CYCLOPROPANATION AS KEY STEP
N. Rosenbaum, Karlsruhe Institute of Technology, Karlsruhe, Germany
FLOW PHOTOCHEMISTRY FOR EFFICIENT AND SCALABLE SYNTHESIS
J.D. Williams, University of Graz, Graz, Austria
APPLICATION OF [2+2+2] CYCLOADDITION IN THE TOTAL SYNTHESIS OF SELAGINPULVILINES
L. Rycek, Charles University of Prague, Prague, Czech Republic
PALLADIUM CATALYZED INTERMOLECULAR IMINE FORMATION
M. Mihelač, University of Ljubljana, Ljubljana, Slovenia
TOTAL SYNTHESIS OF SPHINGOLIPIDS AND SPHINGOSINE-TYPE SIGNALING MOLECULES OF MICROBIAL ORIGIN
L. Raguž, Hans-Knöll Institute (HKI), Jena, Germany
TOWARDS THE TRIARYLATED TRIAZOLIUM SALTS
M. Virant, University of Ljubljana, Ljubljana, Slovenia
CONSECUTIVE INTRAMOLECULAR DEHYDRO-DIELS-ALDER REACTIONS OF HETEROATOM-TETHERED TETRAYNES FOR THE SYNTHESIS OF HETEROLE-CONTAINING POLYCYCLIC COMPOUNDS
A. Sekine, Waseda University, Tokyo, Japan
DEPROTONATIVE GENERATION OF CYCLOALKYNES USING METAL AMIDES
Y. Hioki, Kobe University, Kobe, Japan
SYNTHESIS AND CHARACTERIZATION OF SELENOPHENE-BASED ORGANIC SEMICONDUCTORS
B. Holzer, TU Wien, Vienna, Austria
BENZO[d]THIAZOLE-2-SULFONYL GROUP AS A NITROGEN ACTIVATING AND PROTECTING GROUP
F. Zálešák, Palacky University, Olomouc, Czech Republic
α,β-UNSATURATED α-BENZOTHIAZOLYLSUFONYL DERIVATIVES - PREPARATION AND APPLICATIONS
O. Kováč, Palacky University, Olomouc, Czech Republic
DACH-BASED BIFUNCTIONAL UREA/AMMONIUM SALT CATALYZED ASYMMETRIC α-HYDROXYLATION OF β-KETOESTERS
Ch. Mairhofer, Johannes Kepler University Linz, Linz, Austria
THE SYNTHESIS OF 2,5-DISUBSTITUTED PYRROLES FOR THE INHIBITION OF SOD1 AGGREGATION IN ALS
R. Schirmacher, CBIN Göttingen, Göttingen, Germany
TUNEABLE ACCESS TO MEDICINALLY RELEVANT SCAFFOLDS VIA AN ENANTIOSELECTIVE DEAROMATIVE CYCLISATION CASCADE
J. Rossi-Ashton, University of York, York, UK
USE OF CHROMONE-3-CARBOXYLIC ACID AND ITS DERIVATIVES IN THE SYNTHESIS OF HETEROCYCLES
M. Kornev, The Ural Federal University, Ekaterinburg, Russia
NEW APPROACHES TO SYNTHESIS OF 4H-CHROMENES
V. Osyanin, Samara State Technical University, Samara, Russia
STEREOSELECTIVE SYNTHESIS OF MEDICINALLY-RELEVANT DIHYDROISOQUINOLINONES
M. Amer, University of Bristol, Bristol, UK
SYNTHESIS OF PHOSPHORUS TACRINE ANALOGUES AS A NEW POTENTIAL ANTI-ALZHEIMER'S DISEASE AGENTS
M. Przybyłowska, Gdańsk University of Technology, Gdańsk, Poland
C-H FUNCTIONALIZATION OF N-METHYLATED AMINO ACIDS AND PEPTIDES AS TOOL IN NATURAL PRODUCT SYNTHESIS
T. Kinsinger, Saarland University, Saarbrücken, Germany
MICROWAVE ASSISTED SYNTHESIS OF H-PHOSPHONATES
J.-M. Pohl, Justus Liebig University Giessen, Giessen, Germany
SUPRAMOLECULAR ARHITECTURES SUPPORTED BY CATEMERS OF 2,7-DIPYRIDYLFLUORENE WITH ORTHO-, META- OR PARA- DIIODOTETRAFLUOROBENZENE ISOMERS
L. Pop, "Babes Bolyai" University, Cluj-Napoca, Romania
KETONE ACTIVATION ENABLES METAL-FREE ALPHA-ARYLATION AND ALPHA-OXYAMINATION OF ACETOPHENONES
W. Zawodny, University of Vienna, Vienna, Austria
EN ROUTE TO NEISSERIA MENINGITIDIS SEROGROUP Y FULLY SYNTHETIC VACCINE CANDIDATES
S. Neidig, Ludwig-Maximilians University, Munich, Germany
ALPHA-FLUORONITROALKENES: USEFUL BUILDING BLOCKS FOR THE CONSTRUCTION OF NOVEL FLUORINATED HETEROCYCLES
V. Motornov, N.D. Zelinsky Institute of Organic Chemistry, Moscow, Russia
NEW STUDIES TOWARDS THE TOTAL SYNTHESIS OF GULMIRECIN B
A. Paul, University of Tübingen, Tübingen, Germany
MANGANESE CATALYZED ALKYLATION OF AMIDES AND ESTERS
Y.-K. Jang, RWTH Aachen University, Aachen, Germany
BORON DIRECTED, Ni-CATALYZED REDUCTIVE COUPLING OF UNACTIVATED ALKYL AND ARYL HALIDES WITH INTERNAL ALKENES
S. Bera, Ecole Polytechnique Federale de Lausanne (EPFL), Lausanne, Switzerland
SYNTHESIS OF C-1 ALKYNYL TETRAHYDROISOQUINOLINE DERIVATIVES THROUGH THE A3 REDOX-NEUTRAL COUPLING USING COPPER-CATALYSIS AND PHOTOCATALYSIS
M. Ortiz, Universidad Industrial de Santander, Piedecuesta, Colombia
CO2-DERIVED CARBONATES AND POLYCARBONATES TO METHANOL AND DIOLS VIA METAL LIGAND COOPERATIVE CATALYSIS
V. Zubar, RWTH Aachen University, Aachen, Germany
DESIGN, SYNTHESIS AND EVALUATION OF NOVEL INHIBITORS OF KYNURENINE AMINOTRANSFERASE II
M. Maryška, University of Chemistry and Technology, Prague, Czech Republic
SYNTHESIS OF A FAMILY OF STAR-SHAPED MOLECULAR GEARS
C. Kammerer, Université de Toulouse, Toulouse, France
MECHANOCHEMICALLY INDUCED SWITCHING OF SPIROPYRANS
J. Tůma, University of Chemistry and Technology, Prague, Czech Republic
NEW POSSIBILITIES OF 3,9-DIAMINOSUBTITUTED PERYLENES CORE EXTENSION VIA DIELS-ALDER CYCLOADDITION TO BAY REGION
A. Kurpanik, University of Silesia, Katowice, Poland
A BONDING EVOLUTION THEORY PERSPECTIVE OF THE aza-SNAr MECHANISM
S. Richter-Morales, Universidad de Chile, Santiago, Chile
SYNTHESIS OF PYRAZOLO[1,5-a]PYRIDINES CONTAINING PHOSPHONATE MOIETY
I. Philippov, Novosibirsk Institute of Organic Chemistry, Novosibirsk, Russia
A POTENTIAL N-HETEROCYCLIC BASED LIQUID ORGANIC HYDROGEN CARRIERS
M. Ra, Korea Research Institute of Chemical Technology, Daejeon, Republic of Korea
SYNTHESIS AND CHARACTERIZATION OF NOVEL PYRENE AND PHENOTHIAZINE BASED BUILDING BLOCKS FOR ORGANIC SOLAR CELLS AND MOLECULAR ELECTRONICS
M.-I. Nan, "Babes Bolyai" University, Cluj-Napoca, Romania
SELECTIVITY OF PYRAZOLOQUINOLINONE DERIVATIVES TOWARDS THE ALPHA1+/BETA1- INTERFACE OF THE GABAA RECEPTOR
B.A. Vega Alanis, TU Wien, Vienna, Austria
ENERGY-COUPLING FACTOR TRANSPORTER, A NOVEL TARGET FOR ANTIBIOTIC DEVELOPMENT
S. Bousis, Saarland University, Saarbrücken, Germany
INVESTIGATION OF ACTIVE DEMETHYLATION OF 5-METHYL-2'-DEOXYCYTIDINE
E. Korytiaková, Ludwig-Maximilians University, Munich, Germany
DIRECT CROSS‐COUPLING OF ALLYLIC C(sp3)−H BONDS WITH ARYL‐ AND VINYLBROMIDES BY COMBINED NICKEL AND VISIBLE‐LIGHT CATALYSIS
L. Huang, RWTH Aachen University, Aachen, Germany
HYDRATIVE AMINOXYLATION OF THIOALKYNES
G. Di Mauro, University of Vienna, Vienna, Austria
ENANTIOSELECTIVE SEQUENTIAL ALDOL CONDENSATION
E. Abdelraheem, Delft University of Technology, Delft, The Netherlands
BIARYL COUPLING OF TETRA(HETERO)ARYL BORATES VIA ELECTROCHEMICAL OXIDATIONS
A. Music, Ludwig-Maximilians University, Munich, Germany
BIOTRANSFORMATIONS EMPLOYING NITRILE HYDROLYZING ENZYMES TOWARDS THE ENANTIOSELECTIVE SYNTHESIS OF β-AMINO ACIDS
T. Mareya, Waterford Institute of Technology, Waterford, Ireland
DONOR-SUBSTITUTED PYRIDOBENZO(BIS)THIAZOLES AS TWO PHOTON ABSORBING FLUOROFORES FOR BIOIMAGING
J. Nociarová, Comenius University Bratislava, Bratislava, Slovakia
COtab: A SIMPLE AND PRACTICAL SETUP FOR Pd-CATALYZED CARBONYLATION CHEMISTRY
H. Collin, Aarhus University, Aarhus, Denmark
ELECTROCHEMICAL TRANSFORMATION OF TETRAORGANO BORATES TOWARDS HIGHLY FUNCTIONALIZED ALKENES
A. Baumann, Ludwig-Maximilians University, Munich, Germany
SYNTHESIS OF FLUORINATED PYRAZOLO[1,5-a]PYRIDINES
A. Vorob'ev, Novosibirsk Institute of Organic Chemistry, Novosibirsk, Russia
IDENTIFICATION OF ONCOGENE CONTROLLED SIALOSIDES
B. Smith, Stanford University, Stanford, USA
METAL-LIGAND CATALYZED HETEROCYCLIZATION OF ALLENIC ALCOHOLS
A. Brzozowska, RWTH Aachen University, Aachen, Germany
BENZOTHIAZOLE ANALOGUES OF BODIPY DYES WITH A QUADRUPOLAR (D-π-A-π-D) ARCHITECTURE FOR BIOIMAGING
M. Smolíček, Comenius University Bratislava, Bratislava, Slovakia
SYNTHESIS OF NITRO DERIVATIVES AND FATTY ACID ESTERS OF RICINOLEIC ACID STARTING FROM CASTOR OIL
G. Koutoulogenis, National and Kapodistrian University of Athens, Athens, Greece
BRØNSTED ACID CATALYZED C-H FUNCTIONALIZATION OF ARYL SULFOXIDES VIA A CHARGE ACCELERATED [3,3]-SIGMATROPIC REARRANGEMENT OF BUTADIENYL SULFONIUM CATION INTERMEDIATES
S. Khan, Indian Institute of Technology Bombay, Mumbai, India
PLANARIZED PYRIDINE-BASED TRIARYLAMINES FOR FUNCTIONAL ORGANIC MATERIALS
Th. Kader, TU Wien, Vienna, Austria
SYNTHESIS OF CURCUMIN HETEROCYCLIC DERIVATIVES
R. Smits, Latvian Institute of Organic Synthesis, Riga, Latvia
RADICAL-MEDIATED DEAROMATIZATION OF INDOLES WITH SULFINATE REAGENTS AND PHOSPITHES FOR THE SYNTHESIS OF FLUORINATED AND PHOSPHONATED SPIROCYCLIC INDOLINES
D. Ryzhakov, Université Paris-Sud, Orsay, France
3,3′ - DISUBSTITUTED THIOGALACTOSIDES AS INHIBITORS OF GALECTINS
T. Vašíček, Academy of Science of the Czech Republic, Prague, Czech Republic
DECARBOXYLATIVE, AMINOCATALYTIC CASCADES IN THE SYNTHESIS OF 3,4-DIHYDROCOUMARINS
A. Albrecht, Lodz University of Technology, Lodz, Poland
PROBING THE REACTIVITY OF α,β-UNSATURATED ACYL AMMONIUM INTERMEDIATES
J. Wu, University of St. Andrews, St. Andrews, UK
UNSYMMETRICAL Mn(I) PNNOP PINCER CATALYSTS FOR HYDROGEN BORROWING REACTIONS
A. Nawara-Hultzsch, University of Vienna, Vienna, Austria
Cp*Ir(III) CATALYZED BRANCH SELECTIVE ALLYLIC AMIDATION OF UNACTIAVTED OLEFINS
J.-H. Ye, Westfälische Wilhelms-Universität Münster, Münster, Germany
INHIBITION OF LYSOSOMAL GLYCOSIDASES BY MULTIMERIC PRESENTATIONS OF PYRROLIDINE-BASED IMINOSUGARS
A.T. Carmona, Universidad de Sevilla, Sevilla, Spain
BUILDING COVALENT MOLECULAR CAPSULES BY THIOL- MICHAEL ADDITION CLICK REACTION
M.D. Perretti, Universidad de La Laguna (ULL), Tenerife, Spain
SYNTHESIS OF ANTHRAQUINONES AS HUMAN PROTEIN KINASE CK2 INHIBITORS
P. López Rojas, Universidad de La Laguna, La Laguna, Spain
SYNTHETIC DERIVATIVES OF PHYTOCANNABINOIDS
L. Mikulu, University of Chemistry and Technology, Prague, Czech Republic
PROCESS FOR OBTAINING LOW AND HIGH BOILING 1-PROPENYL AND BIS(1-PROPENYL) ETHERS AND SULPHIDES TOWARDS RENEWABLE CATALYTIC SYSTEMS
B. Marcol-Szumilas, University of Silesia, Katowice, Poland
REGIO- AND CHEMOSELECTIVE DEPROTECTION OF PRIMARY ACETATES BY ZIRCONIUM HYDRIDES
A. Joosten, Normandie Université, Rouen, France
SYNTHESIS OF BENZOBOROXOLE DERIVATIVES AS RECEPTORS FOR SIALIC ACID
A. Di Pasquale, University of Birmingham, Birmingham, United Kingdom
SYNTHESIS AND CATALYTIC APPLICATIONS OF DENDRIMER-CARBON NANOTUBES HYBRIDS
A. Desmecht, Université Catholique de Louvain (UCL), Louvain-la-Neuve, Belgium
SYNTHESIS OF FLUOROGENIC PROBES FOR STABILIZATION OF SUPEROXIDE DISMUTASE (SOD1)
V. Mrđen Debono, Georg-August-Universität, Göttingen, Germany
RESPONSE SURFACE MODELLING OF MICROWAVE ASSISTED BISCHLER-NAPIERALSKI REACTION: SYNTHESIS OF EUDOSTOMIN H
S. Legøy Årvik, University of Bergen, Bergen, Norway
INVESTIGATING MONOAMINE OXIDASE ISOFORM SELECTIVITY FOR NEUROTRANSMITTER SUBSTRATES THROUGH THE PRODUCTION OF THERMODYNAMIC CYCLES
S. Turega, Sheffield Hallam University, Sheffield, UK
NICLOSAMIDE DERIVATIVES INHIBIT CIP2A AND REACTIVATE TUMOR SUPPRESSOR PROTEIN PHOSPHATASE 2A IN NON-SMALL CELL LUNG CANCER CELLS
K.-Y. Jung, Korea Research Institute of Chemical Technology, Daejeon, Republic of Korea
DIRECT ACCESS TO β-KETONITRILES VIA NICKEL-CATALYZED CARBONYLATIVE COUPLING OF α-BROMONITRILES WITH ALKYLZINC REAGENTS
A.S. Donslund, University of Aarhus, Aarhus, Denmark
SYNTHESIS AND ANTICANCER ACTIVITY OF NOVEL SALICYLAMIDE DERIVATIVES
P. Magar, University of Pardubice, Pardubice, Czech Republic
SYNTHESIS, CHARACTERIZATION AND EVALUATION OF AMINOXY AND IONIZABLE LIPIDS FOR THE MODULAR ASSEMBLY OF LIPID-BASED NANOPARTICLES FOR EFFICIENT DELIVERY OF THERAPEUTIC NUCLEIC ACIDS
D. Bhosale, Veterinary Research Institute, Brno, Czech Republic
NOVEL BUILDING BLOCK TOWARDS HIGHLY FUNCTIONALIZED CYCLOPENTANOID SCAFFOLDS
B. Ryckaert, Ghent University, Ghent, Belgium
TERPHENYL PHOSPHANES: A NEW GENERATION OF LIGAND FOR PALLADIUM-CATALYZED AMINATION OF ARYL HALIDES WITH PRIMARY AND SECONDARY ARYL AMINES
J.-C. Shi, Guangdong University of Petrochemical Technology, Maoming, China
GEMINAL SILICON/BORON BIMETALLOIDS: VERSATILE BUILDING BLOCKS FOR MOLECULAR DIVERSITY
M. Diaz, Universitat Ramon Llull, Barcelona, Spain
TOWARDS IODANE-DIRECTED ITERATIVE C-H ALKYLATION
A. Shafir, The Barcelona Institute of Science and Technology, Tarragona, Spain
IODANE-DIRECTED ORTHO C-H ALLYLATION AS GATEWAY TORWARDS ADDED VALUE CORES
W.W. Chen, Catalonia Institute for Advanced Chemistry, Barcelona, Spain
ENANTIOSELECTIVE SYNTHESIS OF HETEROCYCLIC NUCLEOSIDES THROUGH ASYMMETRIC [3+2] ANNULATION OF α‑PURINE-SUBSTITUTED ACRYLATES WITH NITRONES
Q. Du, Southern University of Science and Technology, Shenzhen, China
TOTAL SYNTHESIS OF MYCOSEROSIC ACID FROM MYCOBACTERIUM TUBERCULOSIS AND THE PHEROMONE FROM MARGARODES PRIESKAENSIS
G. Le Calvez, University of Groningen, Groningen, The Netherlands
HYDROGENATION OF BORYLATED ARENES
D. Moock, Westfälische Wilhelms-Universität Münster, Münster, Germany
SYNTHESIS OF ACYCLIC DIALKYL AMINES VIA BUCHWALD-HARTWIG AMINATION
T. Täufer, Leibniz Institute for Catalysis, Rostock, Germany
TOWARDS THE SYNTHESIS OF (+)-LOPHOTOXIN
O. Hoff, University of Oxford, Oxford, UK
EFFICIENT SYNTHESIS OF SPHINGOLIPID AND SPHINGOSINE-TYPE CHEMICAL MEDIATORS OF MICROBIAL ORIGIN
D. Leichnitz, Hans-Knöll Institute (HKI), Jena, Germany
LIGAND DESIGN IN THE ASYMMETRIC SYNTHESIS OF TERTIARY ALCOHOLS
R. O'Gara, University College Dublin, Dublin, Ireland
APPLICATIONS OF (THIO)OXALAMIDES IN ORGANOCATALYSIS: SYNTHESIS AND ACTIVITY OF OXALIC DERIVATIVES
R. McCarthy, University College Dublin, Dublin, Ireland
COMPUTATIONAL CHEMISTRY AND ORGANIC SYNTHESIS: LET US BUILD A BRIDGE
B. Maryasin, University of Vienna, Vienna, Austria
ENANTIOSELECTIVE SYNTHESIS OF FLUORADENES BY C(sp2)-H ARYLATION AND APPLICATION TO THE SYNTHESIS OF BUCKYBOWLS
D. Savary, University of Basel, Basel, Switzerland
UMPOLUNG MEDIATED CARBOXYLATION OF ALDEHYDES
M. Juhl, University of Copenhagen, Copenhagen, Denmark
PREPARATION OF INDOLENINES VIA NUCLEOPHILIC AROMATIC SUBSTITUTION
J. Roesslein, University of Zurich, Zurich, Switzerland
TOTAL SYNTHESIS OF HUMAN PHASE I STEROID METABOLITES
N. Kratena, TU Wien, Vienna, Austria
MECHANISTIC INVESTIGATIONS INTO CATALYTIC, CAPSULE-MEDIATED ARENE ALLYLATIONS
P. Boaler, The University of Edinburgh, Edinburgh, UK
SYNTHESIS AND CHARACTERIZATION OF NEW HIGHLY FLUORINATED DIAMINES SUITED FOR POLYMERIZATION
P. Šimon, University of Pardubice, Pardubice, Czech Republic
Zn- AND Sm-INDUCED REDUCTIVE REARRANGEMENT OF 2-ACYL-2,3-DIHYDROBENZOFURANS INTO 4H-CHROMENES
D. Osipov, Samara State Technical University, Samara, Russia
THIETES: A NEW PLATFORM FOR MOLECULAR DIVERSIFICATION
F. Reiners, Ludwig-Maximilians University, Munich, Germany
ORGANO PHOTOINDUCED DECARBOXYLATIVE ALKYLATION OF COUMARINS WITH N-(ACYLOXY)PHTHALIMIDE
K.N. Tripathi, Indian Institute of Technology Dehli, New Dehli, India
SYNTHESIS OF PHOTOCAGED CARBOHYDRATES
F. Hogenkamp, Heinrich-Heine-University Düsseldorf, Jülich, Germany
PEG400 AS SOLVENT IN THE SYNTHESIS OF NEW 7-[4-ALKYL OR (HET)ARYL-1H-1,2,3-TRIAZOL-1-YL)THIENO[3,2-b]PYRIDINES BY Cu(I)-CATALYZED AZIDE-ALKYNE CYCLOADDITION
M.-J.R.P. Queiroz, Universidade do Minho, Braga, Portugal
DIRECT TRANSFORMATION OF AMINO ACIDS INTO DIAZIRINES AND 15N2-DIAZIRINES AND THEIR APPLICATION AS HYPERPOLARIZED MARKERS
Th. Glachet, Normandie Université, Caen, France
ASYMMETRIC BRØNSTED ACID-CATALYZED FRIEDEL‒CRAFTS REACTION OF CYCLIC N-SULFIMINES AND SULFAMIDATES WITH INDOLES
S.-G. Kim, Kyonggi University, Suwon, Republic of Korea
SYNTHESIS OF BENZISOTHIAZOLE DERIVATIVES AS POSSIBLE HIV-1 NUCLEOCAPSID PROTEIN-7 (NCp7) INHIBITORS
C. Muhanji, The Technical University of Kenya, Nairobi, Kenya
PALLADIUM-CATALYSED SYNTHESIS OF MULTIFUNCTIONAL ALKENYL SULFONYL FLUORIDES
T.S.-B. Lou, University of Oxford, Oxford, UK
Pd(0)-CATALYZED DIRECT INTER- AND INTRAMOLECULAR C2 OR C5-H FUNCTIONALIZATION OF 4-CARBOXYIMIDAZOLES
S. Frippiat, Normandie Université, Rouen, France
SYNTHESIS AND EVALUATION OF THE LARVICIDAL ACTIVITY OF THE DERIVATIVES OF THE CINNAMIC ACID IN THE COMBAT TO AEDES AEGYPTI
D. Lima, Federal University of Alagoas
SYNTHESIS OF BODIPY HETERODIMER FORMED BY HYDROGEN BONDING FOR ELECTRONIC TRANSFER INVESTIGATIONS
M. Cordaro, Università di Messina, Messina, Italy
SMALL SCALE COMPOUND ISOLATION USING MASS DIRECTED PURIFICATION
E.S.E. van Beelen, Waters Corporation, Milford, USA
CHIRAL BUILDING BLOCKS IN THE TOTAL SYNTHESIS OF MONOTERPENE INDOLE ALKALOIDS
S. Varga, Hungarian Academy of Sciences, Budapest, Hungary
TETRAALKYLAMMONIUM SALTS AS SURROGATES FOR OLEFINS IN C-H ACTIVATION
D. Schönbauer, TU Wien, Vienna, Austria
RECENT DEVELOPMENTS IN BIOCATALYTIC REDOX REACTIONS
F. Mutti, University of Amsterdam, Amsterdam, The Netherlands
RUTHENIUM-CATALYZED REDUCTIVE ARYLATION OF N-(2-PYRIDINYL)AMIDES WITH ISOPROPANOL AND ARYLBORONATE ESTERS
E. Renders, University of Antwerp, Antwerpen, Belgium
SYNTHESIS OF SPIRO- γ-HYDROXYLACTAM OXINDOLES AS HYBRID PROHIBITIN-2 LIGANDS
S. Ederwish, University of Strasbourg, Strasbourg, France
SYNTHESIS AND BIOLOGICAL EVALUATION OF THE PRECURSOR OF RADIOACTIVE IODINELABELED BIOACTIVE COMPOUND
T. Farkas, PROGRESSIO Engineering Bureau Ltd., Budapest, Hungary
Si-SUBSTITUTED XANTHENE FLUORESCENT DYES WITH NEAR-INFRARED EMISSION
Z. Kaleta, PROGRESSIO Engineering Bureau Ltd., Budapest, Hungary
AMINO-IMIDAZOLONES AS NOVEL CHELATORS FOR METAL IONS: SYNTHESIS, SOLUTION POTENTIOMETRIC STUDY
R. Tabti, University of Strasbourg, Strasbourg, France
THE DOUBLE REDUCTION OF CYCLIC BENZO-FUSED SULFONAMIDES
A. Khalifa, University College Dublin, Dublin, Ireland
SYNTHESIS OF BENZO-FUSED NEOLIGNANS AS POTENTIAL ANTI-INFLAMMATORY AGENTS
T. Dao-Huy, Hanoi University of Science and Technology, Hanoi, Vietnam
ALTERNATING RADICAL STABILITIES. A CONVERGENT ROUTE TO TERMINAL AND INTERNAL BORONATES
J. Michalland, Ecole Polytechnique, Palaiseau, France
ORGANOCATALYTIC HIGHLY ENANTIOSELECTIVE VINYLOGOUS ALDOL REACTION: RAPID ACCESS TO δ-QUARTERNARY α-HYDROXYPHOSPHONATO-3-ALKYLIDENE-2-OXINDOLES
M.K. Jaiswal, Indian Institute of Technology Dehli, New Dehli, India
UMPOLUING ALKYLATION BASED ON THE OXIDATION OF YNAMIDES
S. Shin, Hanyang University, Seoul, Republic of Korea
SYNTHESIS, CHARACTERIZATION AND REACTIVITY OF Pt(II) PCP PINCER COMPLEXES
M. Urlep, University of Ljubljana, Ljubljana, Slovenia
SYNTHESIS, CHARACTERIZATION AND APPLICATION OF NOVEL FULLERENE DERIVATIVES IN PEROVSKITE SOLAR CELLS
K. Misztal, Saule Research Institute Foundation, Wroclaw, Poland
THIOL-ENE CLICK LIGATION AS AN EFFICIENT APPROACH FOR PEPTIDE MACROCYCLIZATION
P. Milbeo, Trinity College Dublin, Dublin, Ireland
ONE-POT SYNTHESIS OF DIAZANAPHTHALENE DIMERS AND TRIMERS VIA C-H SUBSTITUTION
A. Dastan, Atatürk University, Erzurum, Turkey
ASYMMETRIC PHOTOCATALYTIC C-H FUNCTIONALIZATION OF TOLUENE AND DERIVATIVES
D. Mazzarella, Institut Català d’Investigació Química (ICIQ), Tarragona, Spain
FROM RENEWABLE TO USABLE - BIOTRANSFORMATION FROM CARVONE TO CARVOLACTONE AND ITS COPOLYMERISATION WITH LACTIDE
E. Zukic, TU Wien, Vienna, Austria
BORYLATION OF THIOPHENES DRIVEN BY PHOTOCATALYST-FREE VISIBLE LIGHT
R. Pérez-Ruiz, Universitat Politécnica de València, València, Spain
CINCHONA AND BODIPY: AN APPEALING CATALYTIC STRATEGY FOR CHIMIOSELECTIVE PHOTOOXYGENATION
J. Fischer, Université de Nantes, Nantes, France
LATE-STAGE DIVERSIFICATION THROUGH MANGANESE-CATALYZED C−H ACTIVATION: ACCESS TO ACYCLIC, HYBRID, AND STAPLED PEPTIDES
N. Kaplaneris, Georg-August-Universität, Göttingen, Germany
TOWARDS THE TOTAL SYNTHESIS OF ELISABETHIN A
M. Kaiser, TU Wien, Vienna, Austria
GOLD NANOPARTICLE-CATALYZED SILABORATION OF CYCLOPROPYL ALDEHYDES FORMING REARRANGED SILYLOXY BORONATES
M. Stratakis, University of Crete, Heraklion, Greece
LARGAZOLE, A PROMISING SCAFFOLD FOR HDAC INHIBITORS
M. Borgini, University of Siena, Siena, Italy
SYNTHESIS AND STRUCTURE-BASED STUDIES OF FMN RIBOSWITCH LIGANDS: EXPLORING FMN RIBOSWITCH TARGET TO FIND NEW ANTIBIOTICS
Muhammad, University of Bergen, Bergen, Norway
IMIDAZO[1,2‐c]PYRIMIDIN‐5(6H)‐ONE AS A NOVEL CORE OF CYCLINDEPENDENT KINASE 2 INHIBITORS
A. Lycka, Research Institute for Organic Syntheses (VUOS), Pardubice, Czech Republic
NOVEL APPROACH TO HETEROCYCLES BY TRANSITION METAL CATALYZED [2+2+2] CYCLOADDTIONS
T. Glaesel, Johannes Kepler University Linz, Linz, Austria
DIASTEREO- AND ENANTIOPURE HELICENE 2,2'-BIPYRIDINES: A NEW TYPE OF CHIROPTICAL SWITCHES
I.G. Stará, Czech Academy of Sciences, Prague, Czech Republic
FLUOROFUNCTIONALIZATION OF METAL CORROLES
D. Krisch, Johannes Kepler University Linz, Linz, Austria
C-H ACTIVATION ENABLES A CONCISE AND STEREOSELECTIVE TOTAL SYNTHESIS OF QUININE AND ANALOGUES
M. Berger, University of Vienna, Vienna, Austria
DIRECTED ENANTIOSELECTIVE COUPLING OF ALDEHYDES AND ALKENES
A. Preinfalk, University of Vienna, Vienna, Austria
TANDEM PALLADIUM-CATALYZED INTRAMOLECULAR ADDITION OF ACTIVE METHYLENE COMPOUNDS TO ALKYNES FOLLOWED BY COUPLING WITH (HETERO)ARYL BROMIDES
A. Błocka, Polish Academy of Science, Warsaw, Poland
STEREODIVERGENT SYNTHESIS OF 1,4-DICARBONYLS VIA A TRACELESS SULFOXIDE REARRANGEMENT
I. Klose, University of Vienna, Vienna, Austria
STUDIES ON THE Ru-CATALYZED CARBONYLATIVE MURAI REACTION
G. Poli, Sorbonne Universités, Paris, France
RESOURCE ECONOMY BY COBALTAELECTROCATALYSIS: MERGING ELECTROCHEMISTRY AND C–H ACTIVATION
T.H. Meyer, Georg-August-Universität, Göttingen, Germany
BROMINATION OF 1,2-DISUBSTITUTED CYCLOBUTENES
T. Edlová, University of Chemistry and Technology, Prague, Czech Republic
ASYMMETRIC [3,3]-SIGMATROPIC REARRANGEMENT IN GOLD(I)-CATALYZED INTERMOLECULAR CARBOALKOXYLATION
J. Jang, Hanyang University, Seoul, Republic of Korea
PHOTOBINDING OF TRIFLUSAL TO HUMAN SERUM ALBUMIN INVESTIGATED BY FLUORESCENCE, PROTEOMIC ANALYSIS AND COMPUTATIONAL STUDIES
M.c. Jiménez, Universitat Politécnica de València, València, Spain
A SHORT SEMISYNTHESIS OF HEDERAGONIC ACID BY C–H ACTIVATION
Ch. Knittl-Frank, University of Vienna, Vienna, Austria
OVERCOMING METALLO-β-LACTAMASE MEDIATED RESISTANCE IN BACTERIA
O.A.H. Åstrand, University of Oslo, Oslo, Norway
TOWARDS THE SYNTHESIS OF SAMROIYOTMYCINS A & B
Y.F.A. See, Nanyang Technological University, Singapore
Pd-CATALYZED REDUCTIVE CARBOPERFLUOROALKYLATION OF ALKYNES WITH PERFLUOROALKYL AND ARYL IODIDES VIA BOROPERFLUOROALKYLATION
W. Chaładaj, Polish Academy of Science, Warsaw, Poland
A UNIFIED APPROACH TO THE CHEMOSELECTIVE α-FUNCTIONALIZATION OF AMIDES
C. Gonçalves, University of Vienna, Vienna, Austria
ANTICANCER PROFILE OF NEWLY SYNTHESIZED B-RAF INHIBITORS POSSESS 5(PYRIMIDIN-4-YL)IMIDAZO[2,1-b]OXAZOLE SCAFFOLD
U. Ammar, Korea Institute of Science and Technology, Seoul, Republic of Korea
PHOTO-MEDIATED INTERMOLECULAR HYDROAMINATION OF ACTIVATED OLEFINS USING UNPROTECTED PRIMARY AMINES
F. El-Hage, Leibniz Institute for Catalysis, Rostock, Germany
Pd-CATALYZED HYDROFORMYLATION USING FORMALDEHYDE AS SYNGAS SURROGATES
B. Palucci, Universitat Rovira i Virgili, Tarragona, Spain
TOWARDS THE TOTAL SYNTHESIS OF EUPHOSALICIN AND PEPLUANIN A - ROUTE TO A HIGHLY OXYGENATED CYCLOPENTANE KEY FRAGMENT
J. Templ, TU Wien, Vienna, Austria
ENANTIOSELECTIVE PHOTOCHEMICAL ORGANOCASCADE CATALYSIS
G. Magagnano, Institut Català d’Investigació Química (ICIQ), Tarragona, Spain
THE EFFECTS OF SFC PREPARATIVE SCALE-UP ON THROUGHPUT, PURITY AND RECOVERY OF AN IMPURITY IN AN API MIXTURE
E.S.E. van Beelen, Waters Corporation, Milford, USA
TANDEM CATALYTIC FORMATION AND ENANTIOSELECTIVE [2,3]-REARRANGEMENT OF FUNCTIONALISED ALLYLIC AMMONIUM YLIDES
J. Bitai, University of St. Andrews, St. Andrews, Scotland
ASYMMETRIC TRANSFER HYDROGENATION OF ENONES VIA COUNTERANION ENHANCED CATALYSIS
F. Scharinger, TU Wien, Vienna, Austria
NOVEL CARBAMATE-BASED P,O-LIGANDS IN ASYMMETRIC ALLYLIC ALKYLATIONS
Á.M. Pálvölgyi, TU Wien, Vienna, Austria
CONTINUOUS TRANSFORMATION OF CARBON DIOXIDE USING SUPPORTED IONIC LIQUIDS
A. Sainz Martinez, TU Wien, Vienna, Austria
CATALYTIC METAL-FREE CROSS-COUPLING OF HETEROAROMATIC N-OXIDES WITH ORGANOSILANES
M. Puthanveedu, Max-Planck-Institute for Molecular Physiology, Dortmund, Germany
THIOL–COORDINATED IODONIUM ION CATALYSIS: A DOMINO SYNTHESIS OF Z-SELECTIVE α,β-DIPHENYLTHIO ENONES FROM EASILY ACCESSIBLE SECONDARY ALCOHOLS
N. Sundaravelu, Indian Institute of Technology Madras, Chennai, India
POTENTIALLY TAUTOMERIC 3-ARYLQUINOLIN-4(1H)-ONES VERSUS 3-ARYLQUINOLIN-4-OLS: sPECTROSCOPIC, DFT AND X-RAY ANALYSES
M. Maluleka, University of South Africa, Florida, South Africa
SYNTHESIS, CHARACTERIZATION, AND APPLICATIONS OF SUPPORTED POLYMERIC IONIC LIQUIDS (SILPS)
A. Sahoo, TU Wien, Vienna, Austria
DESIGN AND REGIOSELECTIVE FUNCTIONALIZATION OF NEW 2,4-SUBSTITUED PYRIDO[1',2':1,5]PYRAZOLO[3,4-d]PYRIMIDINES AND 2,4-SUBSTITUED PYRIDO[1',2':1,5]PYRAZOLO[4,3-d]PYRIMIDINES VIA Pd-CATALYZED SEQUENTIAL ARYLATION
A. Ejjoummany, Université Hassan II de Casablanca, Mohammedia, Maroc
SPECTROSCOPIC DATA TO ASSIST CHEMICAL SYNTHESIS
N. Tonge, Mestrelab Research S.L., Santiago de Compostela, Spain
TOWARDS THE TOTAL SYNTHESIS OF PROVIDENCIN
M. Steinacher, TU Wien, Vienna, Austria
DESIGN OF A SELECTIVE AND TUNABLE RCEYM-HYDROGENATION ONE-POT PROCESS
D.N. Prada Gori, Universidad Nacional de Rosario, Rosario, Argentina
EXPLORING THE ROLE OF BASES IN CARBOXYLATION OF GRIGNARD REAGENTS WITH CO2
Y. Yang, University of Copenhagen, Copenhagen, Denmark
RECENT PROGRESS OF AZAINDOLO[3,2,1-jk]CARBAZOLE BASED DONOR-ACCEPTOR MATERIALS AS POTENTIAL TADF EMITTERS
N. Poremba, TU Wien, Vienna, Austria
SYNTHESIS OF N SUBSTITUTED INDOLO[3,2,1-jk]CARBAZOLE BASED SYSTEMS FOR ORGANIC ELECTRONICS
B. Meindl, TU Wien, Vienna, Austria